Evaluation of in vitro absorption, distribution, metabolism, and excretion and assessment of drug-drug interaction of rucaparib, an orally potent poly(ADP-ribose) polymerase inhibitor
Autor: | Jeri Beltman, Thomas Harding, Mingxiang Liao, Jim J. Xiao, Sarah Jaw-Tsai, Andrew Simmons |
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Rok vydání: | 2020 |
Předmět: |
Pharmacology
biology Health Toxicology and Mutagenesis Poly ADP ribose polymerase General Medicine Metabolism Toxicology 030226 pharmacology & pharmacy Biochemistry Poly (ADP-Ribose) Polymerase Inhibitor In vitro 03 medical and health sciences chemistry.chemical_compound 0302 clinical medicine chemistry 030220 oncology & carcinogenesis PARP inhibitor biology.protein Distribution (pharmacology) Rucaparib Polymerase |
Zdroj: | Xenobiotica. 50:1032-1042 |
ISSN: | 1366-5928 0049-8254 |
Popis: | 1. The absorption, distribution, metabolism, elimination, and drug-drug interaction (DDI) potential of the poly(ADP-ribose) polymerase (PARP) inhibitor rucaparib was characterised in vitro.2. Rucap... |
Databáze: | OpenAIRE |
Externí odkaz: | |
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