Synthesis of N-benzothiazol-2-yl-amides by a copper-catalyzed intramolecular cyclization process

Autor:	Zhijin Lu, Feng Peng, Junfeng Bai, Junke Wang, Juli Jiang, Leyong Wang, Yi Pan
Rok vydání:	2008
Předmět:	Ligand Organic Chemistry Intramolecular cyclization chemistry.chemical_element Biochemistry Copper Combinatorial chemistry chemistry.chemical_compound chemistry Thiourea Scientific method Drug Discovery Copper catalyzed Benzamide
Zdroj:	Tetrahedron Letters. 49:467-470
ISSN:	0040-4039
DOI:	10.1016/j.tetlet.2007.11.100
Popis:	Employing N-(4,5-dihydrooxazol-2-yl)benzamide as novel and efficient ligand, the copper-catalyzed intramolecular cyclization of various substituted 1-acyl-3-(2-bromophenyl)thioureas could be successfully carried out under mild conditions. A variety of N-benzothiazol-2-yl-amides were synthesized in good to excellent yields.
Databáze:	OpenAIRE
Externí odkaz:	https://explore.openaire.eu/search/publication?articleId=doi_________::056ee07f2f238f86350e86229b7979fa https://doi.org/10.1016/j.tetlet.2007.11.100 Zobrazit plný text záznamu Full Text from ScienceDirect