Access to NH-aziridine-2-carboxamides through Davidsen acylimidodicarbonate activation
Autor: | Raivis Žalubovskis, Jekaterīna Ivanova, Boriss Štrumfs |
---|---|
Rok vydání: | 2019 |
Předmět: | |
Zdroj: | Comptes Rendus Chimie. 22:283-293 |
ISSN: | 1631-0748 |
Popis: | Acylimidodicarbonates obtained from aziridine-2-carboxamides through Davidsen bis-Boc activation react with amine nucleophiles under mild conditions to form tertiary aziridine-2-carboxylic acid amides. NH aziridine-2-carboxylic acid amides were obtained by hydrogenolythic deprotection of N-Cbz derivatives. |
Databáze: | OpenAIRE |
Externí odkaz: |