Access to NH-aziridine-2-carboxamides through Davidsen acylimidodicarbonate activation

Autor: Raivis Žalubovskis, Jekaterīna Ivanova, Boriss Štrumfs
Rok vydání: 2019
Předmět:
Zdroj: Comptes Rendus Chimie. 22:283-293
ISSN: 1631-0748
Popis: Acylimidodicarbonates obtained from aziridine-2-carboxamides through Davidsen bis-Boc activation react with amine nucleophiles under mild conditions to form tertiary aziridine-2-carboxylic acid amides. NH aziridine-2-carboxylic acid amides were obtained by hydrogenolythic deprotection of N-Cbz derivatives.
Databáze: OpenAIRE