Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4- or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold

Autor: Wachter, R., Chris de Graaf, Keresztes, C., Vandormael, B., Ballet, S., Toth, G., Rognan, D., Tourwé, D.
Přispěvatelé: Medicinal chemistry, AIMMS
Jazyk: angličtina
Rok vydání: 2011
Zdroj: de Wachter, R, de Graaf, C, Keresztes, C, Vandormael, B, Ballet, S, Toth, G, Rognan, D & Tourwé, D 2011, ' Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4-or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold. ', Journal of Medicinal Chemistry, vol. 54, pp. 3384-3393 .
Journal of Medicinal Chemistry, 54, 3384-3393. American Chemical Society
Vrije Universiteit Amsterdam
ISSN: 0022-2623
Databáze: OpenAIRE