Preparation of Enamides via Palladium-Catalyzed Amidation of Enol Tosylates

Autor: Klapars, A., Campos, K. R., Chen, C.-y., Volante, R. P.
Zdroj: Organic Letters; March 2005, Vol. 7 Issue: 6 p1185-1188, 4p
Abstrakt: A Pd-catalyzed coupling of enol tosylates and amides has been developed. Ligand screening revealed dipf as the most general ligand for this transformation. A variety of enol tosylates were coupled to an array of enamides in 58−97% yield.
Databáze: Supplemental Index