Palladium-catalyzed late-stage mono-aroylation of the fully substituted pyrazoles viaaromatic C–H bond activation
Autor: | Chen, Miao-Miao, Shao, Ling-Yan, Lun, Li-Jun, Wu, Yu-Liang, Fu, Xiao-Pan, Ji, Ya-Fei |
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Zdroj: | Chinese Chemical Letters; March 2019, Vol. 30 Issue: 3 p702-706, 5p |
Abstrakt: | A Pd-catalyzed late-stage aroylation of 4-methyl-1,5-diaryl-1 H-pyrazole-3-carboxylates has been developed viadirect Csp2−H bond activation with exclusive site-selectivity, broad substrate scope and good functional group tolerance. |
Databáze: | Supplemental Index |
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