A straightforward synthesis of α-amino phosphonate monoesters using BroP or TPyClU

Autor: Galéotti, Nathalie, Coste, Jacques, Bedos, Philippe, Jouin, Patrick
Zdroj: Tetrahedron Letters; January 1996, Vol. 37 Issue: 23 p3997-3998, 2p
Abstrakt: Monoesters of N-protected α-amino phosphonic acid were prepared from phosphonic acid using BroP or TPyClU as activating agent. This reaction proceeds with good yield, even with hindered alcohols.
Databáze: Supplemental Index