Use of ( S)- N- tert-butoxycarbonylaziridine-2-carboxylate derivatives for α-amino acid synthesis

Autor: Baldwin, Jack E., Farthing, Christopher N., Russell, Andrew T., Schofield, Christopher J., Spivey, Alan C.
Zdroj: Tetrahedron Letters; January 1996, Vol. 37 Issue: 21 p3761-3764, 4p
Abstrakt: ( S)- tert-Butyl- N- tert-butoxycarbonylaziridine-2-carboxylate and ( S)- tert-butyl- N- tert-butoxycarbonylaziridine-2-carboxamide were synthesised and found to react with copper ‘catalysed’ Grignard reagents to give protected α-amino acids in moderate to good yields.
Databáze: Supplemental Index