3-(1H-Tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): A Partial Agonist of the Nicotinic Acid Receptor, G-Protein Coupled Receptor 109a, with Antilipolytic but No Vasodilatory Activity in Mice.

Autor: Graeme Semple, Philip J. Skinner, Tawfik Gharbaoui, Young-Jun Shin, Jae-Kyu Jung, Martin C. Cherrier, Peter J. Webb, Susan Y. Tamura, P. Douglas Boatman, Carleton R. Sage, Thomas O. Schrader, Ruoping Chen, Steven L. Colletti, James R. Tata, M. Gerard Waters, Kang Cheng, Andrew K. Taggart, Tian-Quan Cai, Ester Carballo-Jane, Dominic P. Behan
Zdroj: Journal of Medicinal Chemistry; Jul2008, Vol. 51 Issue 16, p5101-5108, 8p
Databáze: Supplemental Index