Discovery of Quinazoline-2,4(1H,3H)-dione Derivatives Containing 3-Substituted Piperizines as Potent PARP-1/2 Inhibitors Design, Synthesis, In Vivo Antitumor Activity, and X-ray Crystal Structure Analysis.

Autor: Jie Zhou, Ming Ji, Xiaoyu Wang, Hailong Zhao, Ran Cao, Jing Jin, Yan Li, Xianhong Chen, Li Sheng, Xiaoguang Chen, Bailing Xu
Zdroj: Journal of Medicinal Chemistry; 11/25/2021, Vol. 64 Issue 22, p16711-16730, 20p
Databáze: Supplemental Index