Discovery of EST73502, a Dual μ‑Opioid Receptor Agonist and σ1 Receptor Antagonist Clinical Candidate for the Treatment of Pain.

Autor: García, Mónica, Virgili, Marina, Alonso, Mònica, Alegret, Carles, Farran, Joan, Fernández, Begoña, Bordas, Magda, Pascual, Rosalia, Burgueño, Javier, Vidal-Torres, Alba, Fernández de Henestrosa, Antonio R., Ayet, Eva, Merlos, Manuel, Vela, Jose Miguel, Plata-Salamán, Carlos R., Almansa, Carmen
Zdroj: Journal of Medicinal Chemistry; 12/24/2020, Vol. 63 Issue 24, p15508-15526, 19p
Databáze: Supplemental Index