Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders.

Autor: Pellicciari, Roberto, Passeri, Daniela, De Franco, Francesca, Mostarda, Serena, Filipponi, Paolo, Colliva, Carolina, Gadaleta, Raffaella Maria, Franco, Placido, Carotti, Andrea, Macchiarulo, Antonio, Roda, Aldo, Moschetta, Antonio, Gioiello, Antimo
Zdroj: Journal of Medicinal Chemistry; Oct2016, Vol. 59 Issue 19, p9201-9214, 14p
Databáze: Supplemental Index