Design and Synthesis of Pyridone-Containing 3,4-Dihydroisoquinoline-1(2H)-ones as a Novel Class of Enhancer of Zeste Homolog 2 (EZH2) Inhibitors.

Autor: Pei-Pei Kung, Rui, Eugene, Bergqvist, Simon, Bingham, Patrick, Braganza, John, Collins, Michael, Mei Cui, Diehl, Wade, Dinh, Dac, Fan, Connie, Fantin, Valeria R., Gukasyan, Hovhannes J., Wenyue Hu, Buwen Huang, Kephart, Susan, Krivacic, Cody, Kumpf, Robert A., Li, Gary, Maegley, Karen A., McAlpine, Indrawan
Zdroj: Journal of Medicinal Chemistry; Sep2016, Vol. 59 Issue 18, p8306-8325, 20p
Databáze: Supplemental Index