Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Modulators of the Mediator Complex-Associated Kinases CDK8 and CDK19.

Autor: Mallinger, Aurélie, Schiemann, Kai, Rink, Christian, Stieber, Frank, Calderini, Michel, Crumpler, Simon, Stubbs, Mark, Adeniji-Popoola, Olajumoke, Poeschke, Oliver, Busch, Michael, Czodrowski, Paul, Musil, Djordje, Schwarz, Daniel, Ortiz-Ruiz, Maria-Jesus, Schneider, Richard, Ching Thai, Valenti, Melanie, de Haven Brandon, Alexis, Burke, Rosemary, Workman, Paul
Zdroj: Journal of Medicinal Chemistry; Feb2016, Vol. 59 Issue 3, p1078-1101, 24p
Databáze: Supplemental Index