Structure-BasedOptimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors.

Autor: Paul Bamborough, Chun-wa Chung, RebeccaC. Furze, Paola Grandi, Anne-Marie Michon, Robert J. Sheppard, Heather Barnett, Hawa Diallo, DavidP. Dixon, Clement Douault, Emma J. Jones, Bhumika Karamshi, Darren J. Mitchell, Rab K. Prinjha, Christina Rau, RobertJ. Watson, Thilo Werner, Emmanuel H. Demont
Zdroj: Journal of Medicinal Chemistry; Aug2015, Vol. 58 Issue 15, p6151-6178, 28p
Databáze: Supplemental Index