Structure Guided Lead Generationfor M. tuberculosisThymidylate Kinase (Mtb TMK):Discovery of 3-Cyanopyridoneand 1,6-Naphthyridin-2-one as Potent Inhibitors.

Autor: Naik, Maruti, Raichurkar, Anandkumar, Bandodkar, Balachandra S., Varun, Begur V., Bhat, Shantika, Kalkhambkar, Rajesh, Murugan, Kannan, Menon, Rani, Bhat, Jyothi, Paul, Beena, Iyer, Harini, Hussein, Syeed, Tucker, Julie A., Vogtherr, Martin, Embrey, Kevin J., McMiken, Helen, Prasad, Swati, Gill, Adrian, Ugarkar, Bheemarao G., Venkatraman, Janani
Zdroj: Journal of Medicinal Chemistry; Jan2015, Vol. 58 Issue 2, p753-766, 14p
Databáze: Supplemental Index