Discovery of Selective andOrally Bioavailable ProteinKinase Cθ (PKCθ) Inhibitors from a Fragment Hit.

Autor: George, Dawn M., Breinlinger, Eric C., Friedman, Michael, Zhang, Yang, Wang, Jianfei, Argiriadi, Maria, Bansal-Pakala, Pratima, Barth, Martine, Duignan, David B., Honore, Prisca, Lang, Qing Yu, Mittelstadt, Scott, Potin, Dominique, Rundell, Lian, Edmunds, Jeremy J.
Zdroj: Journal of Medicinal Chemistry; Jan2015, Vol. 58 Issue 1, p222-236, 15p
Databáze: Supplemental Index