Synthesis of Substituted 1 H-Indazoles by Pyrazole Annelation to an Arene.

Autor: Garkushenko, A., Sorokina, O., Kryuchkova, G., Zmeev, A., Makarova, M., Vorontsova, M., Sagitullina, G.
Předmět:
Zdroj: Chemistry of Heterocyclic Compounds; May2013, Vol. 49 Issue 2, p273-280, 8p, 2 Charts
Abstrakt: Substituted 1 H-indazoles have been synthesized by reductive intramolecular heterocyclization of 2,4-di-aroyl- N-nitrosomethylanilines and 2,4-diacetyl- N-nitrosomethylaniline. The N-nitrosoanilines were obtained by nitrosation of N-methyl-2,4-diaroyl- and 2,4-diacetylanilines, the products of quaternary 3,5-diaroyl- and 3,5-diacetylpyridinium salt recyclization. [ABSTRACT FROM AUTHOR]
Databáze: Complementary Index