Synthesis of 5-Substituted 1H-Tetrazoles from Aldoximes Using Diphenyl Phosphorazidate.

Autor: Kotaro Ishihara, Mayumi Kawashima, Takayuki Shioiri, Masato Matsugi
Předmět:
Zdroj: Synlett; 2016, Vol. 27 Issue 15, p2225-2228, 4p
Abstrakt: A novel method for the synthesis of 5-substituted 1H-tetrazoles using diphenyl phosphorazidate (DPPA) has been developed. Aromatic and aliphatic aldoximes underwent cycloaddition to afford the corresponding 5-substituted 1H-tetrazoles with ease and efficiency. [ABSTRACT FROM AUTHOR]
Databáze: Complementary Index