| Autor: |
Loreau, Olivier, Camus, Nathalie, Taran, Frédéric, Audisio, Davide |
| Předmět: |
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| Zdroj: |
Synlett; 2016, Vol. 27 Issue 12, p1798-1802, 5p |
| Abstrakt: |
A convenient one-pot synthetic access to 2-aminobenzoxazoles and 2-aminobenzothiazoles has been developed. The protocol uses KCN as starting material and proceeds through an in situ polarity inversion step. This approach provides a new valuable and straightforward entry to carbon-14-radiolabeled pharmaceutically relevant heterocycles and substantially reduces as well the amount of radioactive wastes generated. [ABSTRACT FROM AUTHOR] |
| Databáze: |
Complementary Index |
| Externí odkaz: |
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