A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes.
Autor: | Baud, Matthias G. J.1,2,3, Lin-Shiao, Enrique1,2,4, Cardote, Teresa1, Tallant, Cynthia2,5, Pschibul, Annica1, Kwok-Ho Chan1, Zengerle, Michael1, Garcia, Jordi R.1, Kwan, Terence T.-L.2, Ferguson, Fleur M.2, Ciulli, Alessio1,2 a.ciulli@dundee.ac.uk |
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Zdroj: | Science. 10/31/2014, Vol. 346 Issue 6209, p638-641. 4p. |
Databáze: | Academic Search Ultimate |
Externí odkaz: |