Synthesis and structure–activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor

Autor: Chambers, Laura J. laura.j.chambers@gsk.com, Stevens, Alexander J.1, Moses, Andrew P.1, Michel, Anton D.1, Walter, Daryl S.1, Davies, David J.1, Livermore, David G.1, Fonfria, Elena1, Demont, Emmanuel H.1, Vimal, Mythily1, Theobald, Pam J.1, Beswick, Paul J.1, Gleave, Robert J.1, Roman, Shilina A.1, Senger, Stefan1
Zdroj: Bioorganic & Medicinal Chemistry Letters. May2010, Vol. 20 Issue 10, p3161-3164. 4p.
Databáze: Academic Search Ultimate