Metabolism-driven in vitro/in vivo disconnect of an oral ERɑ VHL-PROTAC.

Autor: Hayhow, Thomas G.1 (AUTHOR) thomas.hayhow@astrazeneca.com, Williamson, Beth1 (AUTHOR), Lawson, Mandy1 (AUTHOR), Cureton, Natalie1 (AUTHOR), Braybrooke, Erin L.1 (AUTHOR), Campbell, Andrew2 (AUTHOR), Carbajo, Rodrigo J.1 (AUTHOR), Cheraghchi-Bashi, Azadeh1 (AUTHOR), Chiarparin, Elisabetta1 (AUTHOR), Diène, Coura R.1 (AUTHOR), Fallan, Charlene1 (AUTHOR), Fisher, David I.3 (AUTHOR), Goldberg, Frederick W.1 (AUTHOR), Hopcroft, Lorna1 (AUTHOR), Hopcroft, Philip3 (AUTHOR), Jackson, Anne3 (AUTHOR), Kettle, Jason G.1 (AUTHOR), Klinowska, Teresa1 (AUTHOR), Künzel, Ulrike3 (AUTHOR), Lamont, Gillian1 (AUTHOR)
Zdroj: Communications Biology. 5/13/2024, Vol. 7 Issue 1, p1-17. 17p.
Databáze: Academic Search Ultimate
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