Design of selective COX-2 inhibitors in the (aza)indazole series. Chemistry, in vitro studies, radiochemistry and evaluations in rats of a [18F] PET tracer.

Autor: Elie, Jonathan1,2 (AUTHOR), Vercouillie, Johnny2,3,4,5 (AUTHOR), Arlicot, Nicolas2,3,4,5 (AUTHOR) nicolas.arlicot@univ-tours.fr, Lemaire, Lucas1 (AUTHOR), Bidault, Rudy2 (AUTHOR), Bodard, Sylvie2 (AUTHOR), Hosselet, Christel2,3 (AUTHOR), Deloye, Jean-Bernard3,6 (AUTHOR), Chalon, Sylvie2 (AUTHOR), Emond, Patrick2 (AUTHOR), Guilloteau, Denis2,3,4,5 (AUTHOR), Buron, Frédéric1 (AUTHOR) frederic.buron@univ-orleans.fr, Routier, Sylvain1 (AUTHOR) frederic.buron@univ-orleans.fr
Zdroj: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2019, Vol. 34 Issue 1, p1-7. 7p.
Databáze: Academic Search Ultimate
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