LUF7244, an allosteric modulator/activator of Kv 11.1 channels, counteracts dofetilide-induced torsades de pointes arrhythmia in the chronic atrioventricular block dog model.

Autor: Qile, Muge1 (AUTHOR), Beekman, Henriette D.M.1 (AUTHOR), Sprenkeler, David J.1 (AUTHOR), Houtman, Marien J.C.1 (AUTHOR), Ham, Willem B.1,2 (AUTHOR), Stary‐Weinzinger, Anna2 (AUTHOR), Beyl, Stanislav2 (AUTHOR), Hering, Steffen2 (AUTHOR), Berg, Dirk‐Jan3 (AUTHOR), Lange, Elizabeth C.M.3 (AUTHOR), Heitman, Laura H.4 (AUTHOR), IJzerman, Ad P.4 (AUTHOR), Vos, Marc A.1 (AUTHOR), Heyden, Marcel A.G.1 (AUTHOR) m.a.g.vanderheyden@umcutrecht.nl, van Ham, Willem B5,6 (AUTHOR), Stary-Weinzinger, Anna6 (AUTHOR), van den Berg, Dirk-Jan7 (AUTHOR), de Lange, Elizabeth C M7 (AUTHOR), van der Heyden, Marcel A G5 (AUTHOR)
Zdroj: British Journal of Pharmacology. Oct2019, Vol. 176 Issue 19, p3871-3885. 15p. 1 Diagram, 2 Charts, 6 Graphs.
Databáze: Academic Search Ultimate
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