Discovery of a series of 8-(1-phenylpyrrolidin-2-yl)-6-carboxamide-2-morpholino-4H-chromen-4-one as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours
Autor: | Barlaam, Bernard, Cosulich, Sabina, Degorce, Sébastien, Ellston, Rebecca, Fitzek, Martina, Green, Stephen, Hancox, Urs, Lambert-van der Brempt, Christine, Lohmann, Jean-Jacques, Maudet, Mickaël, Morgentin, Rémy, Plé, Patrick, Ward, Lara, Warin, Nicolas |
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Zdroj: | In Bioorganic & Medicinal Chemistry Letters 1 May 2017 27(9):1949-1954 |
Databáze: | ScienceDirect |
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