Dehydroevodiamine and hortiamine, alkaloids from the traditional Chinese herbal drug Evodia rutaecarpa, are IKr blockers with proarrhythmic effects in vitro and in vivo.

Autor: Baburin, Igor1 igor.baburin@univie.ac.at, Varkevisser, Rosanne2, Schramm, Anja3, Saxena, Priyanka1, Beyl, Stanislav1, Szkokan, Phillip1,4, Linder, Tobias1, Stary-Weinzinger, Anna1, van der Heyden, Marcel A.G.2, Houtman, Marien2, Takanari, Hiroki2, Jonsson, Malin2, Beekman, Jet H.D.2, Hamburger, Matthias3, Vos, Marc A.2, Hering, Steffen1
Zdroj: Pharmacological Research. May2018, Vol. 131, p150-163. 14p.
Databáze: Academic Search Ultimate