Synthesis and biological evaluation of disubstituted N⁶-cyclopentyladenine analogues: the search for a neutral antagonist with high affinity for the adenosine A1 receptor.

Autor: de Ligt, Rianne A. F.¹, van der Klein, Pieter A. M.¹, von Frijtag Drabbe Künzel, Jacobien K.¹, Lorenzen, Anna², El Maate, Fatna Ait¹, Fujikawa, Shelly¹, van Westhoven, Rosemarijn¹, van den Hoven, Thijs¹, Brussee, Johannes¹, IJzerman, Ad P.¹ ijzerman@lacdr.leidenuniv.nl

Publikováno v: Bioorganic & Medicinal Chemistry. Jan2004, Vol. 12 Issue 1, p139-149. 11p.

Synthesis of 2,3,5-Tri-O-benzyl-D-arabinitol 1,4-Cyclic Sulfate and Its Conversion into Potential Precursors of Shikimate Substrate Analogues

Autor: van der Klein, Pieter A. M., de Nooy, Arjan E. J., van der Marel, Gijs A., van Boom, Jacques H.

Publikováno v: Synthesis; January 1991, Vol. 1991 Issue: 5 p347-349, 3p

Synthesis and biological evaluation of disubstituted N6-cyclopentyladenine analogues: the search for a neutral antagonist with high affinity for the adenosine A1 receptor.

Autor: de Ligt RA; Division of Medicinal Chemistry, Leiden/Amsterdam Center for Drug Research, Leiden University, PO Box 9502, 2300 RA, Leiden, The Netherlands., van der Klein PA, von Frijtag Drabbe Künzel JK, Lorenzen A, Ait El Maate F, Fujikawa S, van Westhoven R, van den Hoven T, Brussee J, IJzerman AP

Publikováno v: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2004 Jan 02; Vol. 12 (1), pp. 139-49.