Zobrazeno 1 - 10
of 85
pro vyhledávání: '"van Westen GJP"'
Publikováno v:
Reference Module in Biomedical Sciences
Drug-induced liver injury (DILI) is one of the prevailing causes of fulminant hepatic failure. It is estimated that three idiosyncratic drug reactions out of four result in liver transplantation or death. Additionally, DILI is the most common reason
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=core_ac_uk__::240b2668dc3d4701639222d502f5b330
https://researchonline.ljmu.ac.uk/id/eprint/12084/1/DILI_review_MS.pdf
https://researchonline.ljmu.ac.uk/id/eprint/12084/1/DILI_review_MS.pdf
Autor:
Ctibor Škuta, Igor V. Tetko, Andreas Bender, Pavel Kříž, Daniel Svozil, G. J. P. van Westen, Wim Dehaen, Isidro Cortes-Ciriano
Publikováno v:
Journal of Cheminformatics, 12, 39
Journal of Cheminformatics
Journal of Cheminformatics, Vol 12, Iss 1, Pp 1-16 (2020)
Journal of Cheminformatics
Journal of Cheminformatics, Vol 12, Iss 1, Pp 1-16 (2020)
Funder: FP7 People: Marie-Curie Actions; doi: http://dx.doi.org/10.13039/100011264; Grant(s): 238701, 238701
An affinity fingerprint is the vector consisting of compound’s affinity or potency against the reference panel of protein targets. Her
An affinity fingerprint is the vector consisting of compound’s affinity or potency against the reference panel of protein targets. Her
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::62c3fe2e04882a74a8c2c7c7bc0110b9
http://hdl.handle.net/1887/106085
http://hdl.handle.net/1887/106085
Autor:
González Hernández MA; Computational Drug Discovery, Leiden Academic Centre for Drug Research, Einsteinweg 55, 2333 CC, Leiden, The Netherlands., Verschuren L; Unit Healthy Living and Work, TNO, The Netherlands Organization for Applied Scientific Research, 2333 BE, Leiden, The Netherlands., Caspers MPM; Unit Healthy Living and Work, TNO, The Netherlands Organization for Applied Scientific Research, 2333 BE, Leiden, The Netherlands., Morrison MC; Unit Healthy Living and Work, TNO, The Netherlands Organization for Applied Scientific Research, 2333 BE, Leiden, The Netherlands., Venhorst J; Unit Healthy Living and Work, TNO, The Netherlands Organization for Applied Scientific Research, 2333 BE, Leiden, The Netherlands., van den Berg JT; Computational Drug Discovery, Leiden Academic Centre for Drug Research, Einsteinweg 55, 2333 CC, Leiden, The Netherlands., Coornaert B; Galapagos NV, 2800, Mechelen, Belgium., Hanemaaijer R; Unit Healthy Living and Work, TNO, The Netherlands Organization for Applied Scientific Research, 2333 BE, Leiden, The Netherlands., van Westen GJP; Computational Drug Discovery, Leiden Academic Centre for Drug Research, Einsteinweg 55, 2333 CC, Leiden, The Netherlands. gerard@lacdr.leidenuniv.nl.
Publikováno v:
Scientific reports [Sci Rep] 2024 Oct 07; Vol. 14 (1), pp. 23362. Date of Electronic Publication: 2024 Oct 07.
Autor:
Dilweg MA; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Mocking TAM; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Maragkoudakis P; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., van Westen GJP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Heitman LH; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl.; Oncode Institute 2333 CC Leiden The Netherlands., IJzerman AP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., Jespers W; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl., van der Es D; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University Einsteinweg 55 2333 CC Leiden The Netherlands d.van.der.es@lacdr.leidenuniv.nl.
Publikováno v:
RSC medicinal chemistry [RSC Med Chem] 2024 Sep 12. Date of Electronic Publication: 2024 Sep 12.
Autor:
den Hollander LS; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Zweemer AJM; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Béquignon OJM; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Hammerl DM; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Bleijs BTM; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Veenhuizen M; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Lantsheer WJF; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Chau B; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., van Westen GJP; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., IJzerman AP; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands., Heitman LH; Leiden Academic Centre for Drug Research, Division of Drug Discovery and Safety, Leiden, the Netherlands; Oncode Institute, the Netherlands. Electronic address: l.h.heitman@lacdr.leidenuniv.nl.
Publikováno v:
Biochemical pharmacology [Biochem Pharmacol] 2024 Aug 05; Vol. 229, pp. 116464. Date of Electronic Publication: 2024 Aug 05.
Autor:
Beerkens BLH; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.; Oncode Institute, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Andrianopoulou V; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Wang X; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Liu R; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., van Westen GJP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Jespers W; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., IJzerman AP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Heitman LH; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.; Oncode Institute, Einsteinweg 55, 2333 CC Leiden, The Netherlands., van der Es D; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
Publikováno v:
ACS chemical biology [ACS Chem Biol] 2024 Jul 19; Vol. 19 (7), pp. 1554-1562. Date of Electronic Publication: 2024 Jun 26.
Autor:
Houvast RD; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands. R.D.Houvast@lumc.nl., Badr N; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., March T; Department of Clinical Pharmacy and Toxicology, Leiden University Medical Center, Leiden, the Netherlands., de Muynck LDAN; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Sier VQ; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Schomann T; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands.; Department of Radiology, Leiden University Medical Center, Leiden, the Netherlands., Bhairosingh S; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Baart VM; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Peeters JAHM; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., van Westen GJP; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden, the Netherlands., Plückthun A; Department of Biochemistry, University of Zürich, Zurich, Switzerland., Burggraaf J; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands.; Centre for Human Drug Research, Leiden, the Netherlands., Kuppen PJK; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Vahrmeijer AL; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands., Sier CFM; Department of Surgery, Leiden University Medical Center, Leiden, the Netherlands.
Publikováno v:
European journal of nuclear medicine and molecular imaging [Eur J Nucl Med Mol Imaging] 2024 Jul; Vol. 51 (8), pp. 2179-2192. Date of Electronic Publication: 2023 Aug 29.
Autor:
Dilweg MA; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., Gorostiola González M; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., de Ruiter MD; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., Meijboom NJ; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., van Veldhoven JPD; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., Liu R; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., Jespers W; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., van Westen GJP; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., Heitman LH; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands.; Oncode Institute, Leiden, The Netherlands., IJzerman AP; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands., van der Es D; Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research, Leiden University, PO Box 9502, Leiden, The Netherlands. d.van.der.es@lacdr.leidenuniv.nl.
Publikováno v:
Purinergic signalling [Purinergic Signal] 2024 Jun 15. Date of Electronic Publication: 2024 Jun 15.
Autor:
van Veggel L; Department of Neuroscience, BIOMED Biomedical Research Institute, Faculty of Medicine and Life Sciences, Hasselt University, 3590 Hasselt, Belgium.; Department of Psychiatry and Neuropsychology, Division of Translational Neuroscience, European Graduate School of Neuroscience, School for Mental Health and Neuroscience, Maastricht University, 6200 Maastricht, The Netherlands.; University MS Center (UMSC), 3900 Hasselt-Pelt, Belgium., Mocking TAM; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Sijben HJ; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Liu R; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Gorostiola González M; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Dilweg MA; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Royakkers J; Sensor Engineering Department, Faculty of Science and Engineering, Maastricht University, 6200 Maastricht, The Netherlands., Li A; Centre for Medicines Discovery, Nuffield Department of Medicine, University of Oxford, OX3 7BN Oxford, U.K., Kumar V; Centre for Medicines Discovery, Nuffield Department of Medicine, University of Oxford, OX3 7BN Oxford, U.K., Dong YY; Nuffield Department of Clinical Neurosciences, Weatherall Institute of Molecular Medicine, University of Oxford, OX3 7BN Oxford, U.K., Bullock A; Centre for Medicines Discovery, Nuffield Department of Medicine, University of Oxford, OX3 7BN Oxford, U.K., Sauer DB; Centre for Medicines Discovery, Nuffield Department of Medicine, University of Oxford, OX3 7BN Oxford, U.K., Diliën H; Sensor Engineering Department, Faculty of Science and Engineering, Maastricht University, 6200 Maastricht, The Netherlands., van Westen GJP; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands., Schreiber R; Section of Psychopharmacology, Neuropsychology and Psychopharmacology, Faculty of Psychology and Neuroscience, Maastricht University, 6200 Maastricht, The Netherlands., Heitman LH; Leiden Academic Centre for Drug Research (LACDR), Division of Drug Discovery and Safety, Leiden University, 2333 Leiden, The Netherlands.; Oncode Institute, Einsteinweg 55, 2333 Leiden, The Netherlands., Vanmierlo T; Department of Neuroscience, BIOMED Biomedical Research Institute, Faculty of Medicine and Life Sciences, Hasselt University, 3590 Hasselt, Belgium.; Department of Psychiatry and Neuropsychology, Division of Translational Neuroscience, European Graduate School of Neuroscience, School for Mental Health and Neuroscience, Maastricht University, 6200 Maastricht, The Netherlands.; University MS Center (UMSC), 3900 Hasselt-Pelt, Belgium.
Publikováno v:
ACS chemical neuroscience [ACS Chem Neurosci] 2024 Apr 03; Vol. 15 (7), pp. 1424-1431. Date of Electronic Publication: 2024 Mar 13.
Autor:
Gorostiola González M; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.; Oncode Institute, 2333 CC Leiden, The Netherlands., Rakers PRJ; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Jespers W; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., IJzerman AP; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands., Heitman LH; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.; Oncode Institute, 2333 CC Leiden, The Netherlands., van Westen GJP; Leiden Academic Centre of Drug Research, Leiden University, Einsteinweg 55, 2333 CC Leiden, The Netherlands.
Publikováno v:
International journal of molecular sciences [Int J Mol Sci] 2024 Mar 26; Vol. 25 (7). Date of Electronic Publication: 2024 Mar 26.