Zobrazeno 1 - 10
of 36
pro vyhledávání: '"da Silva Dadda A"'
Autor:
Paz, Josiane Delgado, Denise de Moura Sperotto, Nathalia, Ramos, Alessandro Silva, Pissinate, Kenia, da Silva Rodrigues Junior, Valnês, Abbadi, Bruno Lopes, Borsoi, Ana Flávia, Rambo, Raoní Scheibler, Corso Minotto, Ana Carolina, da Silva Dadda, Adilio, Galina, Luiza, Macchi Hopf, Fernanda Souza, Muniz, Mauro Neves, Borges Martinelli, Leonardo Kras, Roth, Candida Deves, Madeira Silva, Rodrigo Braccini, Perelló, Marcia Alberton, de Matos Czeczot, Alexia, Neves, Christiano Ev, Duarte, Lovaine Silva, Leyser, Mariana, Dias de Oliveira, Sílvia, Bizarro, Cristiano Valim, Machado, Pablo, Basso, Luiz Augusto
Publikováno v:
In European Journal of Medicinal Chemistry 5 January 2023 245 Part 1
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Sperotto, Nathalia D. de Moura, Silva, Rodrigo Braccini Madeira, Perelló, Marcia Alberton, Borsoi, Ana Flávia, da Silva Dadda, Adilio, Roth, Candida Deves, Freitas, Raquel Dal Sasso, de Souza, Ana Paula Duarte, Freitas, Deise do Nascimento de, Picada, Jaqueline Nascimento, de Sousa, Jayne Torres, Nabinger, Débora Dreher, Altenhofen, Stefani, Bonan, Carla Denise, Rodrigues-Junior, Valnês S., Bizarro, Cristiano Valim, Basso, Luiz Augusto, Machado, Pablo
Publikováno v:
In Biomedicine & Pharmacotherapy July 2021 139
Autor:
Nathalia D. de Moura Sperotto, Rodrigo Braccini Madeira Silva, Marcia Alberton Perelló, Ana Flávia Borsoi, Adilio da Silva Dadda, Candida Deves Roth, Raquel Dal Sasso Freitas, Ana Paula Duarte de Souza, Deise do Nascimento de Freitas, Jaqueline Nascimento Picada, Jayne Torres de Sousa, Débora Dreher Nabinger, Stefani Altenhofen, Carla Denise Bonan, Valnês S. Rodrigues-Junior, Cristiano Valim Bizarro, Luiz Augusto Basso, Pablo Machado
Publikováno v:
Biomedicine & Pharmacotherapy, Vol 139, Iss , Pp 111672- (2021)
Human thymidine phosphorylase (hTP) is overexpressed in several solid tumors and is commonly associated with aggressiveness and unfavorable prognosis. 6-(((1,3-Dihydroxypropan-2-yl)amino)methyl)-5-iodopyrimidine-2,4(1H,3H)-dione (CPBMF-223) is a nonc
Externí odkaz:
https://doaj.org/article/6974146b079f4acc9c3fe70b9fb77449
Autor:
Macchi, Fernanda Souza, Pissinate, Kenia, Villela, Anne Drumond, Abbadi, Bruno Lopes, Rodrigues-Junior, Valnês, Nabinger, Débora Dreher, Altenhofen, Stefani, Sperotto, Nathalia, da Silva Dadda, Adílio, Subtil, Fernanda Teixeira, de Freitas, Talita Freitas, Erhart Rauber, Ana Paula, Borsoi, Ana Flávia, Bonan, Carla Denise, Bizarro, Cristiano Valim, Basso, Luiz Augusto, Santos, Diógenes Santiago, Machado, Pablo
Publikováno v:
In European Journal of Medicinal Chemistry 15 July 2018 155:153-164
Autor:
Bruno L. Abbadi, Valnês da Silva Rodrigues-Junior, Adilio da Silva Dadda, Kenia Pissinate, Anne D. Villela, Maria M. Campos, Luiz G. de França Lopes, Cristiano V. Bizarro, Pablo Machado, Eduardo H. S. Sousa, Luiz A. Basso
Publikováno v:
Frontiers in Microbiology, Vol 9 (2018)
The emergence of strains of Mycobacterium tuberculosis resistant to isoniazid (INH) has underscored the need for the development of new anti-tuberculosis agents. INH is activated by the mycobacterial katG-encoded catalase-peroxidase, forming an acylp
Externí odkaz:
https://doaj.org/article/49524d1e299f4d0a85b2af687585d918
Autor:
Ana Flávia Borsoi, Laura Manzoli Alice, Nathalia Sperotto, Alessandro Silva Ramos, Bruno Lopes Abbadi, Fernanda Souza Macchi Hopf, Adilio da Silva Dadda, Raoní S. Rambo, Rodrigo Braccini Madeira Silva, Josiane Delgado Paz, Kenia Pissinate, Mauro Neves Muniz, Christiano Ev Neves, Luiza Galina, Laura Calle González, Marcia Alberton Perelló, Alexia de Matos Czeczot, Mariana Leyser, Sílvia Dias de Oliveira, Graziela de Araújo Lock, Bibiana Verlindo de Araújo, Teresa Dalla Costa, Cristiano Valim Bizarro, Luiz Augusto Basso, Pablo Machado
Publikováno v:
ACS medicinal chemistry letters. 13(8)
Using cycloalkyl and electron-donating groups to decrease the carbonyl electrophilicity, a novel series of 2-(quinoline-4-yloxy)acetamides was synthesized and evaluated as
Autor:
Josiane Delgado Paz, Nathalia Denise de Moura Sperotto, Alessandro Silva Ramos, Kenia Pissinate, Valnês da Silva Rodrigues Junior, Bruno Lopes Abbadi, Ana Flávia Borsoi, Raoní Scheibler Rambo, Ana Carolina Corso Minotto, Adilio da Silva Dadda, Luiza Galina, Fernanda Souza Macchi Hopf, Mauro Neves Muniz, Leonardo Kras Borges Martinelli, Candida Deves Roth, Rodrigo Braccini Madeira Silva, Marcia Alberton Perelló, Alexia de Matos Czeczot, Christiano Ev Neves, Lovaine Silva Duarte, Mariana Leyser, Sílvia Dias de Oliveira, Cristiano Valim Bizarro, Pablo Machado, Luiz Augusto Basso
Publikováno v:
European Journal of Medicinal Chemistry. 245:114908
Herein a series of 4-aminoquinolines were synthesized in an attempt to optimize and study the structural features related to LABIO-17 biological activity, a Mycobacterium tuberculosis NADH-dependent enoyl-acyl carrier protein reductase (MtInhA) inhib
Autor:
Bruno L. Abaddi, Adilio da Silva Dadda, Luiz Augusto, Etienne C. Waldow, Raoní S. Rambo, Maiele D. Silveira, Nathalia D. M. Sperotto, Pablo Machado, Cristiano Valim Bizarro
Publikováno v:
Journal of the Brazilian Chemical Society, Volume: 32, Issue: 7, Pages: 1413-1423, Published: 02 JUL 2021
Journal of the Brazilian Chemical Society v.32 n.7 2021
Journal of the Brazilian Chemical Society
Sociedade Brasileira de Química (SBQ)
instacron:SBQ
Journal of the Brazilian Chemical Society v.32 n.7 2021
Journal of the Brazilian Chemical Society
Sociedade Brasileira de Química (SBQ)
instacron:SBQ
Using molecular simplification and molecular hybridization approaches, a series of 2-(benzylthio)-1H-benzo[d]imidazoles was synthesized and evaluated as in vitro inhibitors of Mycobacterium tuberculosis (M. tuberculosis) growth. Compounds 6p and 6z w
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::92da5933de3995dd0aceafbe3b4bf11a
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0103-50532021000701413&lng=en&tlng=en
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0103-50532021000701413&lng=en&tlng=en
Autor:
Fávero Reisdorfer Paula, Adilio da Silva Dadda, Diógenes Santiago Santos, Cristiano Valim Bizarro, Pedro Bergo, Nathalia D. M. Sperotto, Maria M. Campos, Fernanda Souza Macchi, Candida Deves Roth, Sidnei Moura, Talita Freitas de Freitas, Luiz Augusto Basso, Christiano Ev Neves, Valnês S. Rodrigues-Junior, Pablo Machado, Ana Paula de Souza
Publikováno v:
Journal of Medicinal Chemistry. 62:1231-1245
Overexpressed human thymidine phosphorylase (hTP) has been associated with cancer aggressiveness and poor prognosis by triggering proangiogenic and antiapoptotic signaling. Designed as transition-state analogues by mimicking the oxacarbenium ion, nov