Zobrazeno 1 - 10
of 140
pro vyhledávání: '"butyrylcholinesterase inhibition"'
Autor:
Gulia Bikbaeva, Anna Pilip, Anastasia Egorova, Ilya Kolesnikov, Dmitrii Pankin, Kirill Laptinskiy, Alexey Vervald, Tatiana Dolenko, Gerd Leuchs, Alina Manshina
Publikováno v:
Nanomaterials, Vol 13, Iss 17, p 2409 (2023)
Photopharmacology is a booming research area requiring a new generation of agents possessing simultaneous functions of photoswitching and pharmacophore. It is important that any practical implementation of photopharmacology ideally requires spatial c
Externí odkaz:
https://doaj.org/article/c56f9f185e4d4f7e84f5beef64bb7ee4
Akademický článek
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Publikováno v:
Molecules, Vol 26, Iss 4, p 989 (2021)
Based on the broad spectrum of biological activity of hydrazide–hydrazones, trifluoromethyl compounds, and clinical usage of cholinesterase inhibitors, we investigated hydrazones obtained from 4-(trifluoromethyl)benzohydrazide and various benzaldeh
Externí odkaz:
https://doaj.org/article/279c19a6ab754560a19480f1e7bf4271
Autor:
Martin Krátký, Zsuzsa Baranyai, Šárka Štěpánková, Katarína Svrčková, Markéta Švarcová, Jiřina Stolaříková, Lilla Horváth, Szilvia Bősze, Jarmila Vinšová
Publikováno v:
Molecules, Vol 25, Iss 10, p 2268 (2020)
Based on the isosterism concept, we have designed and synthesized homologous N-alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides (from C1 to C18) as potential antimicrobial agents and enzyme inhibitors. They were obtained from 4-(trifluoro
Externí odkaz:
https://doaj.org/article/3c6d6b176c1346e4b2467b3b3616f90b
Akademický článek
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Autor:
Jarmila Vinšová, Martin Krátký, Markéta Komlóová, Echchukattula Dadapeer, Šárka Štěpánková, Katarína Vorčáková, Jiřina Stolaříková
Publikováno v:
Molecules, Vol 19, Iss 6, Pp 7152-7168 (2014)
A new series of 27 diethyl 2-(phenylcarbamoyl)phenyl phosphorothioates (thiophosphates) was synthesized, characterized by NMR, IR and CHN analyses and evaluated against Mycobacterium tuberculosis H37Rv, Mycobacterium avium and two strains of Mycobact
Externí odkaz:
https://doaj.org/article/61e6a30b8749480ba20de41b367501d3
Publikováno v:
Volume: 43, Issue: 4 1170-1182
Turkish Journal of Chemistry
Turkish Journal of Chemistry
Alzheimer's disease (AD) is a progressive neurodegenerative disorder and the main cause of dementia in the elderly population. Since the treatment of AD has been associated with the activity of acetylcholinesterase (AChE) and butyrylcholinesterase (B
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::041512e9d3b2059db566aeb5e84f4cf4
https://doi.org/10.3906/kim-1903-74
https://doi.org/10.3906/kim-1903-74
Publikováno v:
Molecules, Vol 16, Iss 9, Pp 7565-7582 (2011)
A series of novel and highly active acetylcholinesterase and butyrylcholinesterase inhibitors derived from substituted benzothiazoles containing an imidazolidine-2,4,5-trione moiety were synthesized and characterized. The molecular structure of 1-(2,
Externí odkaz:
https://doaj.org/article/4cfd34fbaa064d9d98bb605a8d0aef58
Publikováno v:
Molecules, Vol 26, Iss 989, p 989 (2021)
Molecules
Volume 26
Issue 4
Molecules
Volume 26
Issue 4
Based on the broad spectrum of biological activity of hydrazide–hydrazones, trifluoromethyl compounds, and clinical usage of cholinesterase inhibitors, we investigated hydrazones obtained from 4-(trifluoromethyl)benzohydrazide and various benzaldeh
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::954fea1a89f64d2516cb6cfa16d0d45c
https://pubmed.ncbi.nlm.nih.gov/33668452
https://pubmed.ncbi.nlm.nih.gov/33668452
Autor:
Kratky, Martin, Baranyai, Zsuzsa, Štěpánková, Šárka, Svrčková, Katarína, Svarcova, Marketa, Stolarikova, Jirina, Horvath, Lilla, Bosze, Szilvia, Vinsova, Jarmila
Publikováno v:
Molecules, Vol 25, Iss 2268, p 2268 (2020)
Molecules
Volume 25
Issue 10
Molecules
Volume 25
Issue 10
Based on the isosterism concept, we have designed and synthesized homologous N-alkyl-2-[4-(trifluoromethyl)benzoyl]hydrazine-1-carboxamides (from C1 to C18) as potential antimicrobial agents and enzyme inhibitors. They were obtained from 4-(trifluoro
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::d6b5752262b4dc16fb7dd639e473d73d
https://www.mdpi.com/1420-3049/25/10/2268
https://www.mdpi.com/1420-3049/25/10/2268