Zobrazeno 1 - 10
of 64
pro vyhledávání: '"butacaine"'
Autor:
Lucia Tamborini, Daniele Betti, Francesca Annunziata, Andrea Pinto, Martina Letizia Contente, Francesco Molinari, Cecilia Pinna
Publikováno v:
Catalysts, Vol 10, Iss 939, p 939 (2020)
Catalysts
Volume 10
Issue 8
Catalysts
Volume 10
Issue 8
A flow-based chemo-enzymatic synthesis of selected APIs (i.e., butacaine, procaine and procainamide) has been developed. A bioreactor made of MsAcT, a versatile acyltransferase from Mycobacterium smegmatis, immobilised on glyoxyl&ndash
garose, w
garose, w
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd19625daa97d0f3b6bfb88429ed7230
https://www.mdpi.com/2073-4344/10/8/939
https://www.mdpi.com/2073-4344/10/8/939
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 139:763-771
Quantum mechanical (QM) calculations were carried out in order to study the host-guest inclusion complexes of procaine hydrochloride (Pro-H) and butacaine hydrochloride (But-H) with α- and β-cyclodextrins (α- and β-CDs) by PM3 and AM1 methods. Th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e2ab12cbe864b8f4f100a6c668c9ef93
https://doi.org/10.1007/s00706-007-0822-z
https://doi.org/10.1007/s00706-007-0822-z
Publikováno v:
European Journal of Pharmaceutical Sciences. 33:29-41
This study of sparingly soluble model drugs assesses (a) how pH and the aqueous boundary layer factors may affect in vitro and in vivo absorption, (b) to what extent single excipients (sodium taurocholate, hydroxypropyl-beta-cyclodextrin, KCl, propyl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::001814ab7347369dea1e7f65971cfd4b
https://doi.org/10.1016/j.ejps.2007.09.009
https://doi.org/10.1016/j.ejps.2007.09.009
Publikováno v:
Pharmaceutical Research. 24:530-545
This study assessed the effect of excipients (sodium taurocholate, 2-hydroxypropyl-β-cyclodextrin, potassium chloride, propylene glycol, 1-methyl-2-pyrrolidone, and polyethylene glycol 400) on the apparent intrinsic solubility properties of eight sp
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::48d750df4e0d7311a539cbf474cf50d6
https://doi.org/10.1007/s11095-006-9169-0
https://doi.org/10.1007/s11095-006-9169-0
Autor:
H S Hendrickson, M C E van Dam-Mieras
Publikováno v:
Journal of Lipid Research, Vol 17, Iss 4, Pp 399-405 (1976)
Using quantitative data previously reported for the penetration of local anesthetics into lecithin monolayers, the effects of surface and subphase concentrations of anesthetics on the inhibition of pancreatic phospholipase A2 action on didecanoyl pho
Externí odkaz:
https://doaj.org/article/680ac46e87604a5282ef15eb007e35e2
Autor:
H S Hendrickson
Publikováno v:
Journal of Lipid Research, Vol 17, Iss 4, Pp 393-398 (1976)
The penetration of tetracaine into monolayers of phosphatidylcholine and trioctanoin at different surface pressures, and the penetration of dibucaine, tetracaine, butacaine, lidocaine, and procaine into monolayers of didecanoylphosphatidylcholine at
Externí odkaz:
https://doaj.org/article/eec4a89c338b4629a236423303c234be
Publikováno v:
Applied and Environmental Microbiology. 61:4334-4342
Corynebacterium glutamicum can be triggered to excrete glutamate by the addition of local anesthetics, particularly tetracaine. Glutamate efflux is a carrier-mediated process and not due to unspecific membrane permeabilization. The concentration of l
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8085e84905a67b8f57f351fbb23d1057
https://doi.org/10.1128/aem.61.12.4334-4342.1995
https://doi.org/10.1128/aem.61.12.4334-4342.1995
Publikováno v:
Analytica Chimica Acta. 303:137-142
The analytical possibilities of the Chemiluminescence observed from some local anaesthetics on acidic permanganate treatment are investigated. Five drugs belonging to the p-aminobenzoate series gave significant emission and the reagent concentrations
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::537245f09b1a1e6f128c1fcf37924217
https://doi.org/10.1016/0003-2670(94)00517-p
https://doi.org/10.1016/0003-2670(94)00517-p
Publikováno v:
Journal of Biological Chemistry. 268:13791-13798
Cyclosporin A (CyA) and L-carnitine (LC) prevented the killing of cultured hepatocytes by anoxia and rotenone but not by cyanide. Neither CyA nor LC affected the rate or extent of the loss of the mitochondrial membrane potential or the rate or extent
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d9986398db74b3fd5121f605ac9b835d
https://doi.org/10.1016/s0021-9258(19)85172-4
https://doi.org/10.1016/s0021-9258(19)85172-4
Autor:
Terry Bridal, David D. Busath
Publikováno v:
Biochimica et Biophysica Acta (BBA) - Biomembranes. 1107:31-38
Ondrias et al. ((1986) Stud. Biophys. 115, 17-22) found that dibucaine, butacaine, and tetracaine reduce the conductance of membranes containing multiple (greater than 10(6)) gramicidin channels. Similar experiments with local anesthetics (LA's) adde
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd2dc040b1bc43944ac04328ba4a1ecd
https://doi.org/10.1016/0005-2736(92)90325-g
https://doi.org/10.1016/0005-2736(92)90325-g