Zobrazeno 1 - 5
of 5
pro vyhledávání: '"and Timothy C. Walsgrove"'
Publikováno v:
Organic Process Research & Development. 3:60-63
Palladium-catalysed aminocarbonylation of a 7-bromo- or 7-iodo-1,4-benzodiazepine with N-Cbz-4,4‘-bipiperidine hydrochloride efficiently introduced the 7-(4,4‘-bipiperidinylcarbonyl) moiety of (2S)...
Autor:
Alan Negus, M. Whiter, and Timothy C. Walsgrove, Simon Howie, John D. Hayler, Paul Oxley, Giles Robert Gordon
Publikováno v:
Organic Process Research & Development. 2:3-9
Two plant syntheses of ropinirole {4-[2-(di-n-propylamino)ethyl]-1,3-dihydro-2H-indolin-2-one hydrochloride, SK&F-101468-A} using the ferric chloride mediated cyclisation of β-nitrostyrenes to form...
Autor:
and Timothy C. Walsgrove, Clive J. Moores, Richard Neville Saunders, Jerome F. Hayes, Richard J. Atkins, Lynne P. Crawford, Michael Anthony Harris, Christopher Wicks, Gary F. Breen, Trevor J. Grinter, Andrew C. Share
Publikováno v:
Organic Process Research & Development. 1:185-197
The 3,4,8-trisubstituted quinoline derivatives 2-butyryl-8-methoxy-4-[(2-methylphenyl)amino]quinoline and 3-butyryl-8-(2-hydroxyethoxy)-4-[(2-methylphenyl)amino]quinoline were prepared using five novel synthetic strategies, each involving a different
Autor:
Timothy C. Walsgrove, Franz Sondheimer
Publikováno v:
Tetrahedron Letters. 19:2719-2722
Publikováno v:
Tetrahedron. 40:4701-4710
A convergent total synthesis of aklavinone, based on the annelation reaction of cyanophthalide addition to an enone as the key step, was accomplished.