Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Zisheng Fan"'
Autor:
Lifan Chen, Zisheng Fan, Jie Chang, Ruirui Yang, Hui Hou, Hao Guo, Yinghui Zhang, Tianbiao Yang, Chenmao Zhou, Qibang Sui, Zhengyang Chen, Chen Zheng, Xinyue Hao, Keke Zhang, Rongrong Cui, Zehong Zhang, Hudson Ma, Yiluan Ding, Naixia Zhang, Xiaojie Lu, Xiaomin Luo, Hualiang Jiang, Sulin Zhang, Mingyue Zheng
Publikováno v:
Nature Communications, Vol 14, Iss 1, Pp 1-21 (2023)
Abstract Drug development based on target proteins has been a successful approach in recent decades. However, the conventional structure-based drug design (SBDD) pipeline is a complex, human-engineered process with multiple independently optimized st
Externí odkaz:
https://doaj.org/article/c4c90579e2754437ac6717ad301ee041
Discovery of ARF1-targeting inhibitor demethylzeylasteral as a potential agent against breast cancer
Autor:
Jie Chang, Ruirui Yang, Lifan Chen, Zisheng Fan, Jingyi Zhou, Hao Guo, Yinghui Zhang, Yadan Liu, Guizhen Zhou, Keke Zhang, Kaixian Chen, Hualiang Jiang, Mingyue Zheng, Sulin Zhang
Publikováno v:
Acta Pharmaceutica Sinica B, Vol 12, Iss 5, Pp 2619-2622 (2022)
Externí odkaz:
https://doaj.org/article/c29ed944a5f84ebd94199f264a44c6a1
Autor:
Xiaolong Wu, Xiaomin Luo, Xiaozhe Wan, Tianbiao Yang, Xiaohong Liu, Feisheng Zhong, Yinghui Zhang, Kaixian Chen, Sulin Zhang, Dingyan Wang, Xutong Li, Ruirui Yang, Zunyun Fu, Zisheng Fan, Mingyue Zheng, Hualiang Jiang
Publikováno v:
Protein & Cell
A fundamental challenge that arises in biomedicine is the need to characterize compounds in a relevant cellular context in order to reveal potential on-target or off-target effects. Recently, the fast accumulation of gene transcriptional profiling da
Autor:
Lifan Chen, Zisheng Fan, Jie Chang, Ruirui Yang, Hao Guo, Yinghui Zhang, Tianbiao Yang, Chenmao Zhou, Zhengyang Chen, Chen Zheng, Xinyue Hao, Keke Zhang, Rongrong Cui, Yiluan Ding, Naixia Zhang, Xiaomin Luo, Hualiang Jiang, Sulin Zhang, Mingyue Zheng
Drug development based on target proteins has been a successful approach in recent decades. A conventional structure-based drug design pipeline is a complex, human-engineered pipeline with multiple independently optimized steps. Advances in end-to-en
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4cd7e30f471740aa45f71c31cde35ca6
https://doi.org/10.1101/2022.03.26.485909
https://doi.org/10.1101/2022.03.26.485909
Autor:
Chuan Zhou, Zisheng Fan, Zehui Zhou, Yupeng Li, Rongrong Cui, Chaoyi Liu, Guizhen Zhou, Xingxing Diao, Hualiang Jiang, Mingyue Zheng, Sulin Zhang, Tianfeng Xu
Publikováno v:
Journal of medicinal chemistry. 65(5)
Regulating SOS1 functions may result in targeted pan-KRAS therapies. Small-molecule SOS1 inhibitors showed promising anticancer potential, and the most advanced inhibitor BI 1701963 is currently under phase I clinical studies. SOS1 agonists provide n
Discovery of ARF1-targeting inhibitor demethylzeylasteral as a potential agent against breast cancer
Autor:
Jie Chang, Ruirui Yang, Lifan Chen, Zisheng Fan, Jingyi Zhou, Hao Guo, Yinghui Zhang, Yadan Liu, Guizhen Zhou, Keke Zhang, Kaixian Chen, Hualiang Jiang, Mingyue Zheng, Sulin Zhang
Publikováno v:
Acta pharmaceutica Sinica. B. 12(5)
Image 1.
Autor:
Xiaoyu Ding, Rongrong Cui, Jie Yu, Tiantian Liu, Tingfei Zhu, Dingyan Wang, Jie Chang, Zisheng Fan, Xiaomeng Liu, Kaixian Chen, Hualiang Jiang, Xutong Li, Xiaomin Luo, Mingyue Zheng
Publikováno v:
Journal of Medicinal Chemistry; 11/25/2021, Vol. 64 Issue 22, p16838-16853, 16p