Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Yulin Chiang"'
Autor:
Yongyi Luo, David M. Fink, Sukhveen Sahni, Guyan Liang, Peter Crackett, Raymond John Boffey, Lee Lan, Magali Mathieu, Jean Merrill, Sam S. Rebello, Bryan Rees, Wei He, Melanie Wong, Thaddeus R. Nieduzak, Jackson Sharon, Yulin Chiang, Nicola Collar, Abdelazize Laoui, Jean-Pierre Guilloteau
Publikováno v:
Bioorganic & Medicinal Chemistry. 13:2723-2739
Inducible nitric oxide synthase (iNOS) has been implicated in various central and peripheral pathophysiological diseases. Our high throughput screening initially identified a weak inhibitor of iNOS, thiocoumarin 13. From this lead, a number of potent
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8462b9b64f53affa7d279cd6d77ae809
https://doi.org/10.1016/j.bmc.2005.02.036
https://doi.org/10.1016/j.bmc.2005.02.036
Autor:
Edward J. Glamkowski, Roy Corbett, Paul G. Conway, Yulin Chiang, Bordeau Kenneth J, Harold B. Hartman, Joseph T. Strupczewski, Mark R. Szewczak, Helsley Grover C, Carole A. Wilmot
Publikováno v:
Journal of Medicinal Chemistry. 38:1119-1131
A series of 3-[[(aryloxy)alkyl]piperidinyl]-1,2-benzisoxazoles was synthesized and evaluated as potential antipsychotic D2/5-HT2 antagonists. Most of these compounds showed potent antipsychotic-like activity in an apomorphine-induced climbing mouse p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f177932202e0f4169412a6f14bfe5e3
https://doi.org/10.1021/jm00007a009
https://doi.org/10.1021/jm00007a009
Publikováno v:
Tetrahedron Letters. 25:487-490
A practical approach to the synthesis of (±) acivicin (1) and (±) bromo-acivicin (6) has been developed. It centers on the synthesis of alkene 10 by a thermal [3,3] sigmatropic rearrangement of trichloroimidate 9.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1aa13a49f259b930aa89aa41855ebff1
https://doi.org/10.1016/s0040-4039(00)99918-0
https://doi.org/10.1016/s0040-4039(00)99918-0
Publikováno v:
Drug Development Research. 11:169-175
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4b86e7478bc2acbb29658cc049f50653
https://doi.org/10.1002/ddr.430110304
https://doi.org/10.1002/ddr.430110304
Autor:
Mark R. Szewczak, Michael L. Cornfeldt, Robert W. Dunn, Jeffrey C. Wilker, Harry M. Geyer, Stuart Fielding, Edward J. Glamkowski, Yulin Chiang
Publikováno v:
Drug Development Research. 11:157-168
HP 370 4,9-Dibromo-6-(4 methyl-1-piperaziny(l)benzo((b)pyrrolo[3,2,1-jk][1,4 benzodiazepine] demonstrated preclinical activity indicative of clinical atypical antipsychotic activity, which may provide an advantage over current therapeutic agents. It
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1dbe31e485b36def313ebfdb13967163
https://doi.org/10.1002/ddr.430110303
https://doi.org/10.1002/ddr.430110303
Publikováno v:
The Journal of Organic Chemistry. 52:5601-5605
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b51196860a1c2704d78e917d0f260c83
https://doi.org/10.1021/jo00234a017
https://doi.org/10.1021/jo00234a017
Publikováno v:
The Journal of Organic Chemistry. 49:2037-2039
Synthese en 4 etapes a partir du butene-2 diol-1,4 via une transposition sigmatrope carboximidate-carboxamide
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::327b736a3f24d1125cf1c8b4b14eeea4
https://doi.org/10.1021/jo00185a049
https://doi.org/10.1021/jo00185a049
Publikováno v:
ChemInform. 19
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3843d720958e52bdca420e7487c9df53
https://doi.org/10.1002/chin.198820295
https://doi.org/10.1002/chin.198820295