Garcinolic Acid Distinguishes Between GACKIX Domains and Modulates Interaction Networks.

Autor: Breen ME; Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Joy ST; Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Baruti OJ; Program in Chemical Biology, Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Beyersdorf MS; Program in Chemical Biology, Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Henley MJ; Program in Chemical Biology, Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., De Salle SN; Program in Chemical Biology, Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Ycas PD; Department of Chemistry, University of Minnesota, 207 Pleasant St SE, Minneapolis, MN-55455, USA., Croskey A; Program in Chemical Biology, Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Cierpicki T; Department of Pathology, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA., Pomerantz WCK; Department of Chemistry, University of Minnesota, 207 Pleasant St SE, Minneapolis, MN-55455, USA., Mapp AK; Department of Chemistry and Life Sciences Institute, University of Michigan, 210 Washtenaw Avenue, Ann Arbor, MI-48109, USA.

Publikováno v: Chembiochem : a European journal of chemical biology [Chembiochem] 2023 Nov 02; Vol. 24 (21), pp. e202300439. Date of Electronic Publication: 2023 Sep 07.

NMR Analyses of Acetylated H2A.Z Isoforms Identify Differential Binding Interactions with the Bromodomain of the NURF Nucleosome Remodeling Complex.

Autor: Olson NM; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Kroc S; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Johnson JA; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Zahid H; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Ycas PD; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Chan A; Drug Discovery Department, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States., Kimbrough JR; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Kalra P; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States., Schönbrunn E; Drug Discovery Department, H. Lee Moffitt Cancer Center and Research Institute, 12902 Magnolia Drive, Tampa, Florida 33612, United States., Pomerantz WCK; Department of Chemistry, University of Minnesota, 207 Pleasant Street Southeast, Minneapolis, Minnesota 55455, United States.

Publikováno v: Biochemistry [Biochemistry] 2020 May 26; Vol. 59 (20), pp. 1871-1880. Date of Electronic Publication: 2020 May 11.

Selectivity, ligand deconstruction, and cellular activity analysis of a BPTF bromodomain inhibitor.

Autor: Kirberger SE; Department of Chemistry, University of Minnesota, 207 Pleasant St. SE., Minneapolis, MN 55455, USA. wcp@umn.edu., Ycas PD, Johnson JA, Chen C, Ciccone MF, Woo RWL, Urick AK, Zahid H, Shi K, Aihara H, McAllister SD, Kashani-Sabet M, Shi J, Dickson A, Dos Santos CO, Pomerantz WCK

Publikováno v: Organic & biomolecular chemistry [Org Biomol Chem] 2019 Feb 13; Vol. 17 (7), pp. 2020-2027.

Meeting Proceedings ICBS2016-Translating the Power of Chemical Biology to Clinical Advances.

Autor: Kuriki Y; Graduate School of Pharmaceutical Sciences, University of Tokyo , 7-3-1, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan., Komatsu T; Graduate School of Pharmaceutical Sciences, University of Tokyo , 7-3-1, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.; Japan Science and Technology Agency (JST) , 4-1-8 Honcho Kawaguchi, Saitama 332-0012, Japan., Ycas PD; Department of Chemistry, University of Minnesota , 312 Smith Hall, 207 Pleasant St. SE, Minneapolis, Minnesota 55455-0431, United States., Coulup SK; Department of Medicinal Chemistry, University of Minnesota , 717 Delaware Street, SE, Minneapolis, Minnesota 55414, United States., Carlson EJ; Department of Medicinal Chemistry, University of Minnesota , 717 Delaware Street, SE, Minneapolis, Minnesota 55414, United States., Pomerantz WCK; Department of Chemistry, University of Minnesota , 312 Smith Hall, 207 Pleasant St. SE, Minneapolis, Minnesota 55455-0431, United States.; Department of Medicinal Chemistry, University of Minnesota , 717 Delaware Street, SE, Minneapolis, Minnesota 55414, United States.

Publikováno v: ACS chemical biology [ACS Chem Biol] 2017 Apr 21; Vol. 12 (4), pp. 869-877. Date of Electronic Publication: 2017 Mar 17.