Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Yayoi Takao"'
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Median survival times in a CFPAC-1 peritoneal dissemination model after S-1, TAS-114, or S-1 and TAS-114 combination treatment
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f60cdf7d0cd216ad12f8c357b4c534c0
https://doi.org/10.1158/1535-7163.22505167
https://doi.org/10.1158/1535-7163.22505167
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
TAS-114 possesses moderate DPD inhibitory activity, and its inhibition mode is reversible
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::658668c85bafdb66537343b28dc9707c
https://doi.org/10.1158/1535-7163.22505185.v1
https://doi.org/10.1158/1535-7163.22505185.v1
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Cytotoxicity effects of 5-FU, FdUrd, and paclitaxel in combination with TAS-114 in various human cancer cell lines
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4e5dabff1151b01da430dbbd986064d6
https://doi.org/10.1158/1535-7163.22505170
https://doi.org/10.1158/1535-7163.22505170
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Pharmacokinetic analysis of S-1 and TAS-114 combination in SD rats
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::37060639c612dda3772086e17e3728c2
https://doi.org/10.1158/1535-7163.22505179.v1
https://doi.org/10.1158/1535-7163.22505179.v1
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Expression levels of dUTPase in various tumor xenografts and antitumor efficacy of S-1 and TAS-114 combination in various xenograft models
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::09ae661327ebd8cc8ab1895762ca9552
https://doi.org/10.1158/1535-7163.22505182
https://doi.org/10.1158/1535-7163.22505182
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Enzyme kinetic analysis of human dUTPase inhibition by TAS-114 and calculation of Km and Ki values
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2dc5af9d0ac38a761b5cf2d2d4858d74
https://doi.org/10.1158/1535-7163.22505188.v1
https://doi.org/10.1158/1535-7163.22505188.v1
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
X-ray crystallography data and refinement statistics
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::29d8479d6796422ca7fb187c480789f3
https://doi.org/10.1158/1535-7163.22505176.v1
https://doi.org/10.1158/1535-7163.22505176.v1
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
5-Fluorouracil (5-FU) is an antimetabolite and exerts antitumor activity via intracellularly and physiologically complicated metabolic pathways. In this study, we designed a novel small molecule inhibitor, TAS-114, which targets the intercellular met
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2485ebfe75b2d4a58266ecd04dde0732
https://doi.org/10.1158/1535-7163.c.6537976.v1
https://doi.org/10.1158/1535-7163.c.6537976.v1
Autor:
Kenichi Matsuo, Masayoshi Fukuoka, Yayoi Takao, Khoon Tee Chong, Junko Taguchi, Hitoshi Miyakoshi, Seiji Miyahara, Eiji Matsushima, Kunihiro Yoshisue, Akio Fujioka, Keisuke Yamamura, Takeshi Wakasa, Tatsushi Yokogawa, Wakako Yano
Detail description of TAS-114 synthesis
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::40b3a7a05af178ac059675ae7a942041
https://doi.org/10.1158/1535-7163.22505191.v1
https://doi.org/10.1158/1535-7163.22505191.v1
Autor:
Tatsushi Yokogawa, Seiji Miyahara, Eiji Matsushima, Yayoi Takao, Takeshi Wakasa, Junko Taguchi, Kenichi Matsuo, Keisuke Yamamura, Khoon Tee Chong, Hitoshi Miyakoshi, Wakako Yano, Masayoshi Fukuoka, Kunihiro Yoshisue, Akio Fujioka
Publikováno v:
Molecular Cancer Therapeutics. 17:1683-1693
5-Fluorouracil (5-FU) is an antimetabolite and exerts antitumor activity via intracellularly and physiologically complicated metabolic pathways. In this study, we designed a novel small molecule inhibitor, TAS-114, which targets the intercellular met