Synthesis, anti-leishmanial and molecular docking study of bis-indole derivatives

Autor: Muhammad Taha, Imad Uddin, Mohammed Gollapalli, Noor Barak Almandil, Fazal Rahim, Rai Khalid Farooq, Muhammad Nawaz, Mohamed Ibrahim, Mohammed A. Alqahtani, Yasser A. Bamarouf, Manikandan Selvaraj

Publikováno v: BMC Chemistry, Vol 13, Iss 1, Pp 1-12 (2019)

Abstract We have synthesized new series of bisindole analogs (1–27), characterized by 1HNMR and HR-EI-MS and evaluated for their anti-leishmanial potential. All compounds showed outstanding inhibitory potential with IC50 values ranging from 0.7 ±

Externí odkaz: https://doaj.org/article/bc5931f9ee484180ba445184e10709c0

Synthesis of Chromen-4-One-Oxadiazole Substituted Analogs as Potent β-Glucuronidase Inhibitors

Autor: Muhammad Taha, Fazal Rahim, Muhammad Ali, Muhammad Naseem Khan, Mohammed A. Alqahtani, Yasser A. Bamarouf, Mohammed Gollapalli, Rai Khalid Farooq, Syed Adnan Ali Shah, Qamar Uddin Ahmed, Zainul Amiruddin Zakaria

Publikováno v: Molecules, Vol 24, Iss 8, p 1528 (2019)

Chromen-4-one substituted oxadiazole analogs 1–19 have been synthesized, characterized and evaluated for β-glucuronidase inhibition. All analogs exhibited a variable degree of β-glucuronidase inhibitory activity with IC50 values ranging in betwee

Externí odkaz: https://doaj.org/article/ce68764a349242e6adc845d8c0d0336d

Sustainable Program Assessment Practices: A Review of the ABET and NCAAA Computer Information Systems Accreditation Process

Autor: Saqib Saeed, Abdullah M. Almuhaideb, Yasser A. Bamarouf, Dina A. Alabaad, Hina Gull, Madeeha Saqib, Sardar Zafar Iqbal, Asiya Abdus Salam

Publikováno v: International Journal of Environmental Research and Public Health, Vol 18, Iss 12691, p 12691 (2021)
International Journal of Environmental Research and Public Health; Volume 18; Issue 23; Pages: 12691
International Journal of Environmental Research and Public Health

Program outcome assessment is a complex process that demands careful planning and resources in order to accurately assess higher-order thinking skills. A well-defined assessment approach provides detailed insights into program weaknesses and leads to

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d55278958ca4f6ac3fd1e5858fa56250
https://www.mdpi.com/1660-4601/18/23/12691

Synthesis of oxadiazole-coupled-thiadiazole derivatives as a potent β-glucuronidase inhibitors and their molecular docking study

Autor: Muhammad Taha, Mohammed A. Alqahtani, Munther Alomari, Fazal Rahim, Syahrul Imran, Mohammed Gollapalli, Yasser A. Bamarouf, Ashik Mosaddik, Abdul Wadood, Nizam Uddin

Publikováno v: Bioorganic & Medicinal Chemistry. 27:3145-3155

A new series of oxadiazole with thiadiazole moiety (6–27) were synthesized, characterized by different spectroscopic techniques and evaluated for β-glucuronidase inhibitory potential. Sixteen analogs such as 6, 7, 8, 9, 10, 12, 13, 14, 17, 18, 20,

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::57068ae7cd52ddc8a231eb7fdb602c41
https://doi.org/10.1016/j.bmc.2019.05.049

Student Outcomes Assessment Methodology for ABET Accreditation: A Case Study of Computer Science and Computer Information Systems Programs

Autor: Sardar Zafar Iqbal, Mohammed A. Alqahtani, Yasser A. Bamarouf, Saqib Saeed, Nasro Min-Allah, Aamir Shafi

Publikováno v: IEEE Access, Vol 7, Pp 13653-13667 (2019)

Acquiring academic accreditation for degree programs is a top priority for universities across the world. This is understandable because accreditation not only leads to better content and delivery of these programs but also allows these institutes to

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::56572797767d9505626cb92860f29d08
https://doi.org/10.1109/access.2019.2894066