Zobrazeno 1 - 10
of 17
pro vyhledávání: '"Yarkova Ma"'
Publikováno v:
Acta Naturae
Europe PubMed Central
Europe PubMed Central
The translocator protein (TSPO) promotes the translocation of cholesterol to the inner mitochondrial membrane and mediates steroid formation. In this study, we first report on a biological evaluation of the dipeptide GD-23 (N-carbobenzoxy-L tryptopha
Publikováno v:
Bioorganicmedicinal chemistry. 23(13)
A series of 1-arylpyrrolo[1,2-a]pyrazine-3-carboxamides were designed and synthesized as 18 kDa translocator protein (TSPO) ligands. Anxiolytic-like activity of compounds was evaluated in the open field test and elevated plus maze test. Compounds 1a
Akademický článek
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Autor:
Kryzhanovskii SA; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia. SAK-538@yandex.ru., Barchukov VV; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia., Tsorin IB; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia., Stolyaruk VN; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia., Vititnova MB; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia., Mokrov GV; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia., Yarkova MA; V. V. Zakusov Research Institute of Pharmacology, Moscow, Russia.
Publikováno v:
Bulletin of experimental biology and medicine [Bull Exp Biol Med] 2024 Jun; Vol. 177 (2), pp. 235-237. Date of Electronic Publication: 2024 Aug 01.
Autor:
Gudasheva TA; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Deeva OA; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Pantileev AS; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Mokrov GV; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Rybina IV; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Yarkova MA; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia., Seredenin SB; Federal State Budgetary Institution 'Zakusov Research Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Baltiyskaya, 8, 125315 Moscow, Russia.
Publikováno v:
Molecules (Basel, Switzerland) [Molecules] 2020 Nov 04; Vol. 25 (21). Date of Electronic Publication: 2020 Nov 04.
Autor:
Deeva OA; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia., Pantileev AS; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia., Rybina IV; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia., Yarkova MA; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia., Gudasheva TA; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia. tata-sosnovka@mail.ru., Seredenin SB; Zakusov Research Institute of Pharmacology, 125315, Moscow, Russia.
Publikováno v:
Doklady. Biochemistry and biophysics [Dokl Biochem Biophys] 2019 May; Vol. 484 (1), pp. 17-20. Date of Electronic Publication: 2019 Apr 22.
Autor:
Gudasheva TA; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation., Deeva OA; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation., Mokrov GV; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation., Dyabina AS; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation., Yarkova MA; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation., Seredenin SB; Federal State Budgetary Institution 'Research Zakusov Institute of Pharmacology' (FSBI 'Zakusov Institute of Pharmacology'), Moscow, Russian Federation.
Publikováno v:
Medicinal chemistry (Shariqah (United Arab Emirates)) [Med Chem] 2019; Vol. 15 (4), pp. 383-399.
Autor:
Gudasheva TA; Zakusov Research Institute of Pharmacology, Russian Academy of Medical Sciences, ul. Baltiiskaya 8, Moscow, 125315, Russia. tata-sosnovka@mail.ru., Deeva OA; Zakusov Research Institute of Pharmacology, Russian Academy of Medical Sciences, ul. Baltiiskaya 8, Moscow, 125315, Russia., Yarkova MA; Zakusov Research Institute of Pharmacology, Russian Academy of Medical Sciences, ul. Baltiiskaya 8, Moscow, 125315, Russia., Seredenin SB; Zakusov Research Institute of Pharmacology, Russian Academy of Medical Sciences, ul. Baltiiskaya 8, Moscow, 125315, Russia.
Publikováno v:
Doklady. Biochemistry and biophysics [Dokl Biochem Biophys] 2016 Jul; Vol. 469 (1), pp. 298-301. Date of Electronic Publication: 2016 Sep 07.
Publikováno v:
Eksperimental'naia i klinicheskaia farmakologiia [Eksp Klin Farmakol] 2016; Vol. 79 (1), pp. 7-11.
Autor:
Povarnina PY; V.V. Zakusov Research Institute of Pharmacology of RAMS, ul. Baltiyskaya, 8, Moscow, 125315, Russia., Yarkov SA; V.V. Zakusov Research Institute of Pharmacology of RAMS, ul. Baltiyskaya, 8, Moscow, 125315, Russia., Gudasheva TA; V.V. Zakusov Research Institute of Pharmacology of RAMS, ul. Baltiyskaya, 8, Moscow, 125315, Russia., Yarkova MA; V.V. Zakusov Research Institute of Pharmacology of RAMS, ul. Baltiyskaya, 8, Moscow, 125315, Russia., Seredenin SB; V.V. Zakusov Research Institute of Pharmacology of RAMS, ul. Baltiyskaya, 8, Moscow, 125315, Russia.
Publikováno v:
Acta naturae [Acta Naturae] 2015 Jul-Sep; Vol. 7 (3), pp. 108-12.