Zobrazeno 1 - 10
of 191
pro vyhledávání: '"Y. V. V. Srikanth"'
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 27:2216-2220
Prostate cancer is the most frequently diagnosed malignancy and the leading cause of cancer related death in men. First line therapy for disseminated disease relies on androgen deprivation, leveraging the addiction of these tumors on androgens for bo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ac4469abea3c8c2eec76e1e93902a23b
https://doi.org/10.1016/j.bmcl.2017.03.030
https://doi.org/10.1016/j.bmcl.2017.03.030
Autor:
Jingsheng Xia, Andréia Cristina Karklin Fontana, William Lester, Y. V. V. Srikanth, Yuhong Fang, Sandhya Kortagere, Ole V. Mortensen, Joseph M. Salvino
Publikováno v:
ACS chemical neuroscience. 9(3)
Dysfunction of excitatory amino acid transporters (EAATs) has been implicated in the pathogenesis of various neurological disorders, such as stroke, brain trauma, epilepsy, and neurodegenerative diseases, among others. EAAT2 is the main subtype respo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f93031eb855ae840e85290572e7bc800
https://pubmed.ncbi.nlm.nih.gov/29140675
https://pubmed.ncbi.nlm.nih.gov/29140675
Autor:
Y. V. V. Srikanth, Jiyoon Lee, Seung Bum Park, Ja Young Koo, Jongmin Park, Sangmi Oh, Hankum Park
Publikováno v:
Chemical communications (Cambridge, England). 52(34)
Herein we report molecular shape-dependent nonspecific labeling of photoaffinity linkers (PLs) in the cellular proteome. Linear PLs have a greater tendency to engage in nonspecific binding than branched PLs. Exploiting this property, we discovered a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b0816df3d5e672501d1f72c55f5c6d6e
https://pubmed.ncbi.nlm.nih.gov/27043101
https://pubmed.ncbi.nlm.nih.gov/27043101
Autor:
Y. V. V. Srikanth, Thokhir Basha Shaik, Ahmed Kamal, Md. Ashraf, Shasi V. Kalivendi, M. Naseer A. Khan
Publikováno v:
Letters in Drug Design & Discovery. 9:242-250
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::162fea934e98fc26a650730ff2c92303
https://doi.org/10.2174/157018012799129774
https://doi.org/10.2174/157018012799129774
Autor:
Ahmed Kamal, A. Lavanya, Y. V. V. Srikanth, M. Janaki Ramaiah, Manika Pal-Bhadra, M. Kashi Reddy, S.N.C.V.L. Pushpavalli, M. Naseer A. Khan, Md. Ashraf
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 22:571-578
A series of bisindole–pyrrolobenzodiazepine conjugates ( 5a – f ) linked through different alkane spacers was prepared and evaluated for their anticancer activity. All compounds exhibited significant anticancer potency and the most potent compoun
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::11a493d2dd7a63d144899c2ec4a3b5e7
https://doi.org/10.1016/j.bmcl.2011.10.080
https://doi.org/10.1016/j.bmcl.2011.10.080
Autor:
Y. V. V. Srikanth, Aarti Juvekar, M. Janaki Ramaiah, Manika Pal-Bhadra, G. Bharath Kumar, Surekha M. Zingde, V. Santosh Reddy, Indira Bag, Ahmed Kamal, Rajender, Subrata Sen, M. Kashi Reddy, S.N.C.V.L. Pushpavalli
Publikováno v:
ChemMedChem. 6:1665-1679
A library of new aryl-substituted naphthalene C8-linked pyrrolo[2,1-c][1,4]benzodiazepine (PBD) conjugates with various linker architectures were designed, synthesized, and evaluated for their anticancer activity against a panel of 11 human cancer ce
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ec6efdc90c3689565e6284f78307f152
https://doi.org/10.1002/cmdc.201100207
https://doi.org/10.1002/cmdc.201100207
Autor:
Y. V. V. Srikanth, A. K. Saxena, Nitasha Suri, Ahmed Kamal, M. Naseer A. Khan, Thokhir Basha Shaik, Md. Ashraf, Shasi V. Kalivendi
Publikováno v:
Medicinal Chemistry. 7:165-172
Two series of compounds (5-14 and 15-23) based on the scaffolds of 2-(1,1-dioxido-4-phenyl-4Hbenzo[e][1,2,4]thiadiazin-3-yl)-N-(4-methoxyphenyl)hydrazinecarboxamide (5) and 2-((4-methoxyphenyl)amino)-10-phenyl-10H-benzo[e][1,2,4]triazolo[1,5-b][1,2,4
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5a28325f4d42062bcbc3a7134528838c
https://doi.org/10.2174/157340611795564259
https://doi.org/10.2174/157340611795564259
Autor:
Zheng, Jiabin1 (AUTHOR), Feng, Huolun1,2 (AUTHOR), Lin, Jiatong1,2 (AUTHOR), Zhou, Jianlong1 (AUTHOR), Xi, Zhihui2 (AUTHOR), Zhang, Yucheng1 (AUTHOR), Ling, Fa1 (AUTHOR), Liu, Yongfeng1 (AUTHOR), Wang, Junjiang1 (AUTHOR), Hou, Tieying3,4 (AUTHOR) sz_houtieying@yeah.net, Xing, Fan5 (AUTHOR) xingfan@gdph.org.cn, Li, Yong1,2 (AUTHOR) liyong@gdph.org.cn
Publikováno v:
Advanced Science. 10/28/2024, Vol. 11 Issue 40, p1-17. 17p.
Autor:
Y. V. V. Srikanth, Nisha Kurian, Subrata Sen, Aarti Juvekar, Surekha M. Zingde, K. Srinivasa Reddy, Ahmed Kamal, M. Naseer A. Khan
Publikováno v:
Bioorganic & Medicinal Chemistry. 16:7804-7810
A series of triazolobenzothiadiazine-pyrrolobenzodiazepine conjugates linked through different alkane spacers have been prepared. These compounds have exhibited significant cytotoxicity against most of the cell lines examined. Compound 5a displays GI
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b8335404f90202cafb2548bf7de91d7e
https://doi.org/10.1016/j.bmc.2008.06.056
https://doi.org/10.1016/j.bmc.2008.06.056
Publikováno v:
Energy Sources, Part A: Recovery, Utilization, and Environmental Effects. 30:1534-1539
Simple and precise methods have been developed for the determination of ethanol in blend petrol using gas chromatography and Fourier transform infrared spectroscopy techniques. The methods can determine a minimum quantity of 1% of alcohol in petrol.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5a73c868a875652d7f77f0f5390bd8aa
https://doi.org/10.1080/15567030701258444
https://doi.org/10.1080/15567030701258444