Zobrazeno 1 - 10
of 26
pro vyhledávání: '"Y. V. Faletrov"'
Autor:
L. A. Varfolomeeva, Y. B. Slonimskiy, N. A. Egorkin, M. E. Minyaev, Y. V. Faletrov, K. M. Boyko, N. N. Sluchanko
Publikováno v:
Crystallography Reports. 67:909-917
Autor:
J. U. Panada, V. A. Klopava, T. A. Kulahava, Y. V. Faletrov, N. S. Frolova, S. V. Koran, E. G. Fomina, V. M. Shkumatov
Publikováno v:
Biochemistry (Moscow), Supplement Series B: Biomedical Chemistry. 16:246-252
Publikováno v:
Proceedings of the National Academy of Sciences of Belarus, Chemical Series. 58:186-190
4-methyl-7-methoxycoumarin (CumOMe) has been synthesized and in silico calculations demonstrated localization of methoxy group within 0.4 nm from Fe ion of hem groups for some structures of human CYP19 & CYP46 as well as CYP152 S. paucimobilis, CYP15
Publikováno v:
Proceedings of the National Academy of Sciences of Belarus, Chemical Series. 58:62-67
Publikováno v:
Proceedings of the National Academy of Sciences of Belarus, Chemical Series. 57:456-462
An effective method of synthesis thiazolo[3,2-a]pyrimidine derivatives was developed and the compounds with n-pentyl or β-acetoxycyclopropyl as well as fluorescent benzo[f]coumarin substituents were obtained with yields 60 % and more. Using computat
Autor:
Veronika S. Karpushenkova, Viktoryia A. Zavalinich, Vladimir M. Shkumatov, Y. V. Faletrov, Anastasia D. Shkredava, Polina S. Yakovets
Publikováno v:
Журнал Белорусского государственного университета: Химия, Iss 2, Pp 25-35 (2021)
Albumin is a globular protein of plasma of mammalian blood participating in transport of hydrophobic metabolites and drugs. Thus, studies devoted to its binding are valuable as a part of evaluation of new potential drugs or fluorescent probes for in
Autor:
N. S. Frolova, Y. V. Faletrov, M. S. Horetski, E. V. Rudaya, E. V. Andrievskaya, Anna Brzostek, K. A. Gilep, Aleksandra S. Falchevskaya, Renata Plocinska, J. V. Panada, Vladimir M. Shkumatov
Publikováno v:
Biochemistry (Moscow), Supplement Series B: Biomedical Chemistry. 15:111-118
Molecular docking of four isoniazid hydrazones including steroids dehydroepiandrosterone, pregnenolone, 16α,17α-epoxypregnenolone, and cholestenone (IDHEA, IPRE, IEP5, ICHN), to mycobacterial cytochromes P450 was performed. The in silico study has
Autor:
Sergei V. Kostjuk, Nikita V. Minaev, Evgenii O. Epifanov, Y. V. Faletrov, Petr Timashev, K. N. Bardakova, Yulia A. Piskun
Publikováno v:
Bulletin of the Russian Academy of Sciences: Physics. 84:1406-1410
Hydrophobic derivatives of the antibacterial drug ciprofloxacin are synthesized and used as photoinitiators of two-photon polymerization. A way of selecting 3D printing parameters and the effect they have on scaffold topography are described for phot
Autor:
Aleksandra S. Falchevskaya, M. S. Horetski, E. V. Rudaya, Anna Brzostek, K. A. Gilep, Vladimir M. Shkumatov, Renata Plocinska, J. V. Panada, N. S. Frolova, Y. V. Faletrov, E. V. Andrievskaya
Publikováno v:
Biomeditsinskaya Khimiya. 66:378-385
Molecular docking of four hydrazones of isoniazid with steroids (dehydroepiandrosterone, pregnenolone, 16α,17α-epoxypregnenolone, cholestenone) - IDHEA, IPRE, IEP5, ICHN, to mycobacterial cytochromes P450 was performed. The in silico study has show
Publikováno v:
Biochemistry (Moscow), Supplement Series B: Biomedical Chemistry. 13:357-363
Four isomeric N-alkynylaminosteroids of the androstane and pregnane series were synthesized and tested in vitro for inhibition of CYP450 17A1 heterologously expressed in transgenic yeast Yarrowia lipolytica. The highest inhibitory activity was observ