Zobrazeno 1 - 10
of 26
pro vyhledávání: '"Xiao Shu He"'
Autor:
Ling Zhou, Xiao-Shu He
Publikováno v:
IOP Conference Series: Materials Science and Engineering. 1043:052020
Copula model has been increasingly used in reliability modeling of correlation systems. In this paper, the static copula model, time-varying copula model and variable structure copula model are compared. Firstly, variable structure copula model is in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a60cc4f45da03fa613cf0430e1ecb40e
https://doi.org/10.1088/1757-899x/1043/5/052020
https://doi.org/10.1088/1757-899x/1043/5/052020
Autor:
Xiao-Shu He, Arnold Brossi
Publikováno v:
Journal of Heterocyclic Chemistry. 28:1741-1746
Nortropinone 5, prepared from 3 by N-demethylation with trichloroethyl chloroformate, followed by deprotection of carbamate 4 with zinc in acetic acid, served as a starting material to prepare the N-protected 6-acetoxy ketones 7 and 9–12, and alcoh
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ebc6c626693852cd9b4f35baaaa44662
https://doi.org/10.1002/jhet.5570280716
https://doi.org/10.1002/jhet.5570280716
Autor:
Hutchison Alan J, Kover Renata X, Robbin Brodbeck, Xiao-Shu He, Andrew Thurkauf, Kevin J. Hodgetts, Andrzej Kieltyka, Stanislaw Rachwal, Xiaoyan Zhang, John R. Peterson, Jan W. F. Wasley, Renee J. Primus, He Zhao
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 12:3105-3109
Optimization of the lead compound 2-[-4-(4-chloro-benzyl)-piperazin-1-yl]-1-(2,3-dihydro-indol-1-yl)-ethanone 1 by systematic structure-activity relation (SAR) studies lead to two potent compounds 2-[-4-(4-chloro-benzyl)-piperazin-1-yl]-1-(2-methy-2,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::eb02ce198fbc302c0f8d14590d286292
https://doi.org/10.1016/s0960-894x(02)00655-8
https://doi.org/10.1016/s0960-894x(02)00655-8
Autor:
Xiao-Shu He, Andrew Thurkauf, Andrzej Kieltyka, Jan W. F. Wasley, Robbin Brodbeck, He Zhao, Diane C. Hoffman, Renee J. Primus
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 12:3111-3115
A series of chiral benzylpiperazinyl-1-(2,3-dihydro-indol-1-yl)ethanone derivatives were prepared and examined for their affinity at dopamine D2 and D4 receptors. Three compounds having D2/D4 affinity ratios approximating that found for the atypical
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5e0fd275bd4e4a19ae2bd12af99f435
https://doi.org/10.1016/s0960-894x(02)00656-x
https://doi.org/10.1016/s0960-894x(02)00656-x
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 7:2399-2402
A series of 3-[(4-arylpiperaz-1-yl)alkylamino]-2H-1,4-benzoxazines were prepared and their affinities for cloned human D2, D3, and D4 dopamine receptor subtypes were measured. This led to the identification of 1a, 1f, and 1g as high affinity selectiv
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a5ba0103dcf458079054d6b148bddb0f
https://doi.org/10.1016/s0960-894x(97)00442-3
https://doi.org/10.1016/s0960-894x(97)00442-3
Autor:
B.R. Zeeberg, M.R. Rayeq, R.C. McRee, Richard C. Reba, Daniel R. Weinberger, K. Rice, Kan Sam Lee, E.I. Cohen, S.F. Boulay, V.K. Sood, Xiao Shu He
Publikováno v:
Applied Radiation and Isotopes. 48:27-35
Radioiodinated (R,S)-IQNB and (R,R)-IQNB are prepared either from a triazene precursor or using an exchange reaction. In both cases the radiochemical yield is low. The product of the exchange reaction also suffers from having a fairly low specific ac
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ee0cfa5d1785004a9883df805cb8d085
https://doi.org/10.1016/s0969-8043(96)00125-x
https://doi.org/10.1016/s0969-8043(96)00125-x
Autor:
Kan Sam Lee, Dorota Matecka, Garry Wong, Brian R. de Costa, Xiao-shu He, Kenner C. Rice, Zi-Qiang Gu, Phil Skolnick
Publikováno v:
Journal of Labelled Compounds and Radiopharmaceuticals. 34:27-32
[123I]tert-Butyl 8-iodo-5,6-dihydro-5-methyl-6-oxo-4H-imidazo [1,5-a][1,4]benzodiazepine 3-carboxylate ([123I]3), a high affinity and selective radioligand for the diazepam insensitive (DI) benzodiazepine receptor was synthesized in 2 steps from tert
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::223621af6e4d19daf1234cb896b94df7
https://doi.org/10.1002/jlcr.2580340105
https://doi.org/10.1002/jlcr.2580340105
Publikováno v:
The Journal of Organic Chemistry. 59:482-485
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6ef1340890a81380b6d6623f371a2feb
https://doi.org/10.1021/jo00081a033
https://doi.org/10.1021/jo00081a033
Publikováno v:
Journal of Medicinal Chemistry. 36:4075-4081
We previously reported (J. Med. Chem. 1993, 36, 1188-1193) that changes to the ring size of the piperidine and cyclohexyl rings of the high-affinity and selective dopamine (DA)-uptake inhibitor 1-[1-(2-benzo[b]thienyl)cyclohexyl]piperidine (BTCP, 2)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8ee8b983c5d9e82ef257b2e0f4d8ef05
https://doi.org/10.1021/jm00077a011
https://doi.org/10.1021/jm00077a011
Autor:
Celia Dominguez, Joannes T. M. Linders, W. D. Bowen, Wanda Williams, B. R. De Costa, Xiao-shu He, Zi Qiang Gu
Publikováno v:
Journal of Medicinal Chemistry. 36:2311-2320
As a continuation of our earlier study (J. Med. Chem. 1992, 35, 4334-4343) we conformationally restricted the sigma-receptor ligand 2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylamine (1) by incorporating it into a series of homolog
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::82e3dca88bf0a00421aa06fdd1f55e6d
https://doi.org/10.1021/jm00068a007
https://doi.org/10.1021/jm00068a007