Zobrazeno 1 - 10
of 23
pro vyhledávání: '"Wolfram Gaida"'
Publikováno v:
Neuropharmacology. 49:1220-1227
Neuropathic pain affects many patients, and treatment today is far from being perfect. Nav1.8 Na(+) channels, which are expressed by small fibre sensory neurons, are promising targets for novel analgesics. Na(+) channel blockers used today, however,
Autor:
Klaus Mendla, Andreas Raschig, Helmut Ensinger, Thomas Weiser, Wolfram Gaida, Takeshi Osugi, Angelo Ceci, Marion Wienrich
Publikováno v:
Drug Development Research. 56:321-334
Since the discovery of muscarinic receptor subtypes, extensive research has been going on attempting to provide treatments for diseases related to malfunctions of cholinergic receptors. In Alzheimer's disease, the prevailing symptomatology is a progr
Autor:
Andreas Raschig, Wolfram Gaida, D. Meier, Rudolf Hammer, Helmut Ensinger, Marion Wienrich, A. Walland
Publikováno v:
Life Sciences. 68:2593-2600
In functional pharmacological assays, talsaclidine has been described as a functionally preferential M1 agonist with full intrinsic activity, and less pronounced effects at M2- and M3 receptors. In accordance with this, cholinomimetic central activat
Autor:
Gerd Schnorrenberg, Heike A. Wieland, Beate Rist, Wolfram Gaida, Annette G. Beck-Sickinger, Leonardo Scapozza, Nikolaus Ingenhoven
Publikováno v:
European Journal of Biochemistry. 247:1019-1028
Several attempts to investigate the bioactive conformation of neuropeptide Y have been made so far. As cyclic peptides are much more rigid than linear ones, we decided to synthesise cyclic analogues of the C-terminal dodekapeptide amide neuropeptide
Autor:
L.J.M. Cross, Madeleine Ennis, Michael Bienert, Wolfram Gaida, E. Krause, Annette G. Beck-Sickinger, Günther Jung
Publikováno v:
British journal of pharmacology, 117(2): 325-332
1. Neuropeptide-induced histamine release is thought to occur via receptor-independent mechanisms, with net charge and lipophilicity being important factors. 2. In this study, the histamine releasing ability of neuropeptide Y (NPY), two C-terminal se
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::521048aac5a0e871364bb9930045bccf
https://repository.publisso.de/resource/frl:6405176
https://repository.publisso.de/resource/frl:6405176
Autor:
Günther Jung, Eric Grouzmann, Eike Hoffmann, Annette G. Beck-Sickinger, Hansjörg Dürr, Wolfram Gaida
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 3:937-942
The prerequisite for Y2-mediated biological activity was elaborated by synthesizing analogs of neuropeptide Y (NPY) 1-4-Ahx-25-36. The finding, that a pronounced hydrophobic segment is required in the C-terminal segment for signal transduction led to
Publikováno v:
Biochemical Society Transactions. 20:847-850
Publikováno v:
Biopolymers. 31:613-619
C-terminal analogues of neuropeptide Y (NPY) of small molecular size have been synthesized. The influence of chain length, single or multiple amino acid substitution, and segment substitutions on receptor binding, pre- and postsynaptic biological act
Autor:
Heike A. Wieland, Gerd Schnorrenberg, Wolfgang Eberlein, Franz Esser, Henri Doods, Horst Dollinger, Wolfhard Engel, Wolfram Gaida, Klaus Rudolf
Publikováno v:
European journal of pharmacology. 384(2-3)
The in vitro biological characterisation of the first potent and selective non-peptide neuropeptide Y Y(2) receptor antagonist, (S)-N(2)-[[1-[2-[4-[(R,S)-5,11-dihydro-6(6h)-oxodibenz[b, e]azepin-11-yl]-1-piperazinyl]-2-oxoethyl] cylopentyl] acetyl]-N
Autor:
F. von Bruchhausen, S. Ebel, A. W. Frahm, E. Hackenthal, Margitta Albinus, Hassan-Fahmy Ali, Syed Laik Ali, Gudrun Amschler, Uwe Amschler, Erwin von Angerer, Peter Barth, Wolfgang Barthel, Kurt Bauer, Andrea Bauer, Jürgen Beckmann, Winfried Beil, Jürgen Beitz, Günther Bellmann, Thorsten Beyrich, Franz Bossle, Helmut Bräunlich, Matthias Bräutigam, Kerstin Brinkmann, Adalbert Brinz, Franz von Bruchhausen, Kay Brune, Axel Büge, Ulrich Bürger, Wolfram Christ, Klaus Daneck, Gerd Dannhardt, Helga Doering, Siegfried Ebel, Kurt Eger, Peter Emig, Thomas Erker, Bernhard Feil, Monika Fett, August Wilhelm Frahm, Margarete Frahm, Klaus-Jürgen Freundt, Wolfram Gaida, Detlef Geffken, Ulrich Geis, Klaus Geldsetzer, Ulrich Gessner, Erika Glusa, Berthold Göber, Margarete Goppelt-Strübe, Wilhelm Gössling, Eberhard Gottwald, Beate Grates, Annette Graul, Sibylle Greiner, Adolf Grisk, Michael Grosam, Jan Gustafsson, Hartmut Gustmann, Jürgen Haas, Axel Haberkorn, Eberhard Hackenthal, Annette Häfner, Boris Haluszczynski, Achim Harder, Susanne Hartmann, Heribert Häusler, Marcus Heidenreich, Gerhard Heinemeyer, Bernd Hempel, Monika Herboth, Klaus Herbrand, Sibylle Hoedt-Schmidt, Wolfgang Hoefke, Hermann Hoffmann, Ute Hoffmann-Schollmayer, Bernhard Hofmann, Ulrike Holzgrabe, Anette Hornberger, Ute Hübner-Steiner, Martin Hug, Wolfgang Ibrom, Walter Janßen, Angela Jördens, Ilmar Jurna, Günther Kaiser, Dieter-Abbo Kalbhen, Petra Kisser, Christoph Klett, Stephanie Klett, Gerd Kobal, Johannes Koehler, Axel Kramer, Birgit Krammer, Gottfried Kreutz, Reinhard Kroker, Markus Kuhn, Norbert Kühn, Dorothea Landsiedel, Andreas Langner, Martina Laudszun, Jochen Lehmann, Marion Sylvia Lehner, Stefan Leiner, Hans Löwe, Johannes Mann, Detlef Manns, Wolfgang Matthiessen, Rainer Maue, Peter Maul, Andreas Maurer, Ralf Mayer, Wolfgang Meindl, Werner Meise, Klaus Menges, Paul Messinger, Hans-Jürgen Mest, Frank Peter Meyer, J. Mollière, Rudolf Morgenstern, Wolfgang Morick, Joachim Mössner, Alfred Müller, Walter E. Müller, Klaus Müller, Christa Müller, Daniel Müller, Michael Neugebauer, Ottmar Neugebauer, Peter Nickel, Peter Nuhn, Bernd Nürnberg, Joachim Oertel, Michael Oettel, Tilmann Ott, Thomas Otzen, Hartmut Oßwald, Peter Pachaly, Helmut Pelzer, Karl-Uwe Petersen, Siegfried Pfeifer, Klaus Pietrzik, Kathrin Pöllath, Olaf Queckenberg, Bernd Raffelsberger, Eberhard Reimann, Jörg Remien, Markus Reuß, Andreas Reymann, Joachim Richter, Peter H. Richter, Hubert Richter, Klaus Rittinghaus, Hans Rommelspacher, Gerhard Rücker, Gerhard Schaefer, Klaus Schaefer, Jutta Schcerer, Helmut Schlager, Hildegard Schleinitz, Wolfgang Schlichter, Gerhard Schmidt, Wolfgang Schmutzler, Johannes Schräder, Thomas Schulz-Schalge, Harald Schütz, Helmut Schwilden, Gisela Skopp, Ulrich Speck, Marcus Spohn, Ralf Stahlmann, Johannes-Peter Stasch, E. Staubli, Jürgen Steinmeyer, Karl-Heinz Stiefvater, Michael Streek, Günther Strippel, Karl-Heinz Surborg, Ulf Sürig, Istvan Szelenyi, Alfred Thomas, Herbert Trampisch, Reinhard Troschütz, Bernard Unterhalt, Eugen J. Verspohl, Sabine Vogel, Franz-Josef Volk, Sven Völkl, Heinz Walther, Horst Weber, Martin Wenzel, Marion Weyandt-Spangenberg, Sandra Wich, Burkhard Wichert, Hilke Winterhoff, Peter Witte, Monika Wolff
Publikováno v:
Hagers Handbuch der Pharmazeutischen Praxis ISBN: 9783642634291
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f10a7661271f3853ec38855a5cc69687
https://doi.org/10.1007/978-3-642-57995-0_1
https://doi.org/10.1007/978-3-642-57995-0_1