Zobrazeno 1 - 10
of 40
pro vyhledávání: '"Wolfgang K.-D. Brill"'
Autor:
Hubert Gstach, Andrew G. Cole, Ian R. Henderson, Baldwin John J, Juerg Zimmermann, Roland E. Dolle, Lan-Ying Qin, James R. Wareing, Wolfgang K.-D. Brill, Axel Metzger, Kurt W. Saionz, Marc-Raleigh Brescia
Publikováno v:
Tetrahedron Letters. 50:7082-7085
An efficient and general synthesis of substituted 2-amino-7,8-dihydropteridin-6(5H)-ones using a combination of solution-phase and solid-phase chemistry is described. Solution-phase chemistry was used to produce two pyrimidine regioisomers that were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::226ff5b78225e18bf164076aa818b1f5
https://doi.org/10.1016/j.tetlet.2009.10.005
https://doi.org/10.1016/j.tetlet.2009.10.005
Publikováno v:
Tetrahedron Letters. 48:3535-3538
The Hinsberg thiophene synthesis was expanded to support bound thioglycolic acid derived synthons, which reacted with arils to give thiophenes in high purity.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::22cd35595ee9c1ad85a8356e06885dfb
https://doi.org/10.1016/j.tetlet.2007.03.111
https://doi.org/10.1016/j.tetlet.2007.03.111
Publikováno v:
Tetrahedron. 62:10223-10236
Oxadiazoles were generated upon a dehydrative cyclization reaction with 2-acyl hydrazides bound to the polymeric support via one of their N atoms using TFAA as a dehydration agent.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4d6f56d41bf209b39f3b6565fe7492f3
https://doi.org/10.1016/j.tet.2006.08.016
https://doi.org/10.1016/j.tet.2006.08.016
Autor:
Wolfgang K.‐D. Brill, Gianluca Papeo
Publikováno v:
Combinatorial Chemistry: From Theory to Application, Volume 26, Second Revised Edition
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::66453f68a2dd67ef8f37e63759947f75
https://doi.org/10.1002/3527607706.ch4
https://doi.org/10.1002/3527607706.ch4
Publikováno v:
Tetrahedron. 60:8561-8577
6-Acylmino-1-alkyl/aryl-4-oxo-1,4-dihydrocinnoline-3-carboxamides were synthesized in parallel from 6-nitro-4-oxo-1,4-dihydrocinnoline-3-carboxylic acid. The latter formed amides with amines bound to polystyrene-based resins via acid-labile linkers.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8196f90676666d2e682e057ba3e515d0
https://doi.org/10.1016/j.tet.2004.06.103
https://doi.org/10.1016/j.tet.2004.06.103
Publikováno v:
Molecular Diversity. 6:43-53
The following paper summarizes our work on compound libraries of 2,6,8-trisubstituted purines. This synthesis route on a polystyrene support begins with 2,6-dichloro purine making extensive use of catalysis. During the synthesis the polymer bound pur
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2c31ae54667ee36c32ad364e6851cd19
https://doi.org/10.1023/a:1024895515316
https://doi.org/10.1023/a:1024895515316
Publikováno v:
Tetrahedron Letters. 42:6515-6518
2,6,8-Trisubstituted purines were synthesized from 2,6-dichloropurine bound to polystyrene-based Rink resin at the N(9) position. Selective successive displacements of the chlorine atoms in the 2- and 6-positions followed. Bromination of C(8) and Sti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fe05c2ad011f47b3ba3bb65b891aa4df
https://doi.org/10.1016/s0040-4039(01)01300-4
https://doi.org/10.1016/s0040-4039(01)01300-4
Publikováno v:
Tetrahedron Letters. 42:6279-6282
Diaminopurines, immobilized on a polymeric support are treated with a charge transfer complex of bromine and lutidine to afford 8-brominated derivatives. An ionic complex of bromine and lutidine did not oxidize the purines. 2,6-Dialkylaminopurines co
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::55e658120eec4e93032ec6c9857bf280
https://doi.org/10.1016/s0040-4039(01)01246-1
https://doi.org/10.1016/s0040-4039(01)01246-1
Publikováno v:
Synlett. 2001:1097-1100
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::16e2acfee0b240d595f8f034a754487c
https://doi.org/10.1055/s-2001-15138
https://doi.org/10.1055/s-2001-15138
Publikováno v:
Synlett. 1998:865-868
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::167859cc19a0d2640f5d225fc9a23b4c
https://doi.org/10.1055/s-1998-1808
https://doi.org/10.1055/s-1998-1808