Zobrazeno 1 - 10
of 142
pro vyhledávání: '"Wilma, Quaglia"'
Autor:
Luca Botticelli, Emanuela Micioni Di Bonaventura, Fabio Del Bello, Gianfabio Giorgioni, Alessandro Piergentili, Wilma Quaglia, Alessandro Bonifazi, Carlo Cifani, Maria Vittoria Micioni Di Bonaventura
Publikováno v:
Pharmacological Research, Vol 195, Iss , Pp 106875- (2023)
Neuromedin U (NMU) is a bioactive peptide produced in the gut and in the brain, with a role in multiple physiological processes. NMU acts by binding and activating two G protein coupled receptors (GPCR), the NMU receptor 1 (NMU-R1), which is predomin
Externí odkaz:
https://doaj.org/article/a5eef850d2c64716b12e4792c1bcf571
Autor:
Cecilia Baldassarri, Gianfabio Giorgioni, Alessandro Piergentili, Wilma Quaglia, Stefano Fontana, Valerio Mammoli, Gabriele Minazzato, Elisa Marangoni, Massimiliano Gasparrini, Leonardo Sorci, Nadia Raffaelli, Loredana Cappellacci, Riccardo Petrelli, Fabio Del Bello
Publikováno v:
Pharmaceuticals, Vol 16, Iss 2, p 189 (2023)
The prevention of nicotinamide adenine dinucleotide (NAD) biosynthesis is considered an attractive therapeutic approach against cancer, considering that tumor cells are characterized by an increased need for NAD to fuel their reprogrammed metabolism.
Externí odkaz:
https://doaj.org/article/23800b1cafb64571a44463c8a8295339
Autor:
Alessandro Bonifazi, Fabio Del Bello, Gianfabio Giorgioni, Alessandro Piergentili, Elizabeth Saab, Luca Botticelli, Carlo Cifani, Emanuela Micioni Di Bonaventura, Maria Vittoria Micioni Di Bonaventura, Wilma Quaglia
Publikováno v:
Medicinal Research Reviews.
Autor:
Gianfabio Giorgioni, Fabio Del Bello, Wilma Quaglia, Luca Botticelli, Carlo Cifani, E. Micioni Di Bonaventura, M. V. Micioni Di Bonaventura, Alessandro Piergentili
Publikováno v:
Journal of Medicinal Chemistry. 65:3098-3118
Ghrelin is an octanoylated peptide acting by the activation of the growth hormone secretagogue receptor, namely, GHS-R1a. The involvement of ghrelin in several physiological processes, including stimulation of food intake, gastric emptying, body ener
Autor:
Luca Botticelli, Emanuela Micioni Di Bonaventura, Fabio Del Bello, Gianfabio Giorgioni, Alessandro Piergentili, Adele Romano, Wilma Quaglia, Carlo Cifani, Maria Vittoria Micioni Di Bonaventura
Publikováno v:
Nutrients, Vol 12, Iss 8, p 2288 (2020)
The dopamine D4 receptor (DRD4) has a predominant expression in the prefrontal cortex (PFC), brain area strictly involved in the modulation of reward processes related to both food and drug consumption. Additionally, the human DRD4 gene is characteri
Externí odkaz:
https://doaj.org/article/29b1f3db9bdc4c76a54e835cd6e251e3
Autor:
Maura Pellei, Luca Bagnarelli, Lorenzo Luciani, Fabio Del Bello, Gianfabio Giorgioni, Alessandro Piergentili, Wilma Quaglia, Michele De Franco, Valentina Gandin, Cristina Marzano, Carlo Santini
Publikováno v:
International Journal of Molecular Sciences, Vol 21, Iss 7, p 2616 (2020)
In the present article, copper(I) complexes of bis(pyrazol-1-yl) carboxylic acid (LH), bis(3,5-dimethylpyrazol-1-yl) carboxylic acid (L2H), and bis(pyrazol-1-yl) acetates conjugated with an N-methyl-d-aspartate (NMDA) receptor antagonist (LNMDA or L2
Externí odkaz:
https://doaj.org/article/d6c0f44eaddc4787ada0b57743e45699
Autor:
Thomas M. Keck, Pegi Pavletić, Giulio Vistoli, Wilma Quaglia, Silvia Gervasoni, Fabio Del Bello, Alessandro Bonifazi, Alessandro Piergentili, Amy Hauck Newman, Gianfabio Giorgioni
Publikováno v:
ACS Chemical Neuroscience. 12:3638-3649
In the search for novel bitopic compounds targeting the dopamine D3 receptor (D3R), the N-(2,3-dichlorophenyl)piperazine nucleus (primary pharmacophore) has been linked to the 6,6- or 5,5-diphenyl-1,4-dioxane-2-carboxamide or the 1,4-benzodioxane-2-c
Autor:
Pegi, Pavletić, Ana, Semeano, Hideaki, Yano, Alessandro, Bonifazi, Gianfabio, Giorgioni, Alessandro, Piergentili, Wilma, Quaglia, Maria Giovanna, Sabbieti, Dimitrios, Agas, Giorgio, Santoni, Roberto, Pallini, Lucia, Ricci-Vitiani, Emanuela, Sabato, Giulio, Vistoli, Fabio, Del Bello
Publikováno v:
Journal of medicinal chemistry. 65(18)
To better understand the role of dopamine D
Autor:
Pegi Pavletić, Ana Semeano, Hideaki Yano, Alessandro Bonifazi, Gianfabio Giorgioni, Alessandro Piergentili, Wilma Quaglia, Maria Giovanna Sabbieti, Dimitrios Agas, Giorgio Santoni, Roberto Pallini, Lucia Ricci-Vitiani, Emanuela Sabato, Giulio Vistoli, Fabio Del Bello
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::268fbae6fc98015af05318031ee31348
http://hdl.handle.net/2434/939471
http://hdl.handle.net/2434/939471
Autor:
Emanuela Micioni Di Bonaventura, Luca Botticelli, Fabio Del Bello, Gianfabio Giorgioni, Alessandro Piergentili, Wilma Quaglia, Adele Romano, Silvana Gaetani, Maria Vittoria Micioni Di Bonaventura, Carlo Cifani
Publikováno v:
Pharmacological research. 185
The melanocortinergic neural circuit, known for its influence on energy expenditure and feeding behavior, also plays a role in stress and stress-induced psychiatric disorders, including anxiety and depression. The major contribution is given by the m