Zobrazeno 1 - 10 of 16 pro vyhledávání: '"William Watters"'
1
Synthesis of carbon-14-labelled peptides
Autor: Jason Syvret, Stuart Jones, Sean L. Kitson, Balasubramaniam Upeandran, Rodney T. Brown, Thomas S. Moody, William Watters, Antonio Dell’Isola
Publikováno v: Journal of Labelled Compounds and Radiopharmaceuticals. 62:713-717
Carbon-14 (14 C)-labelled active pharmaceutical ingredients (APIs) and investigational medicinal products (IMPs) are required for phase 0/I to phase III mass balance and micro-dosing clinical trials. In some cases, this may involve the synthesis of 1
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1bb8d85c90092c600026fe95f481f627
https://doi.org/10.1002/jlcr.3777
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2
Developments in AKP Policy Toward Religion and Homogeneity
Autor: Samuel William Watters
Publikováno v: German Law Journal. 19:351-374
Critics of the Turkish interpretation of secularism,laiklik, describe it as authoritarian and repressive. Indeed, rather than establish state neutrality toward religion,laiklikhistorically entailed state control of Islam, the religion of the vast maj
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::bbbe47554b2b82435cfa2c7e03897b82
https://doi.org/10.1017/s2071832200022720
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3
Synthesis of isotopically labelled [14C]ZT-1 (Debio-9902), [d3]ZT-1 and (−)-[d3]huperzine A, a new generation of acetylcholinesterase inhibitors
Autor: Austin McMordie, William Watters, Sean L. Kitson, Loïc Leman, Jana Cairns, Rodney T. Brown, Judith Marfurt, Victor L. Murrell
Publikováno v: Journal of Labelled Compounds and Radiopharmaceuticals. 54:720-730
A method has been developed for the synthesis of two isotopically labelled forms of a pro-drug of the acetylcholinesterase inhibitor (� )-huperzine A. These labelled compounds, [ 14 C]ZT-1 (Debio-9902) and [d3]ZT-1, were used in clinical studies to
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::6a8f9ff0d9f7213b1a5a712856d87d4c
https://doi.org/10.1002/jlcr.1918
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5
Growth Inhibitory Activity of Extracted Material and Isolated Compounds from the Fruits ofKigelia pinnata
Autor: Zoica Delbederi, David Waugh, Barry McClean, Colin O'Dowd, Hendrik W. Van Den Berg, Paul Armstrong, Stephanie Feutren-Burton, William Watters, Catherine A. Higgins, Tanachat Bell
Publikováno v: Planta Medica. 76:1840-1846
A study of the components of the fruits of Kigelia pinnata was undertaken to identify compounds with potential growth inhibitory activity against human melanoma cells, since extracts from the fruits of this plant have been described in traditional me
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9256c58bc77e4a960f7c5331bb493991
https://doi.org/10.1055/s-0030-1250046
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6
Carbon-14 radiosynthesis of 4-(5-chloro-2-hydroxyphenyl)-3-(2-hydroxyethyl)-6-(trifluoromethyl)-[4-14C]quinolin-2(1H)-one (XEN-D0401), A novel BK channel activator
Autor: William Watters, Fiona Chan, Stuart Jones, Sean L. Kitson, David John Madge
Publikováno v: Journal of Labelled Compounds and Radiopharmaceuticals. 53:140-146
A method has been developed for the carbon-14 radiosynthesis of [14C]XEN-D0401, a 4-(2-hydroxyphenyl)quinolin-2(1H)-one derivative. The radiosynthetic route involves a series of ortho-lithiations directed by both 2-methoxymethyl (MOM) and pivaloyl pr
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::abbc2f105011b09251795c5b76850c90
https://doi.org/10.1002/jlcr.1740
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7
Synthesis and in Vitro and in Vivo Evaluation of a Series of Dihydroisocoumarin Derivatives Conjugated with Fatty Acids, Alcohols, and Amines as Potential Anticancer Agents
Autor: Catherine A. Higgins, Paul Armstrong, David Waugh, Zoica Delbederi, Patrick G. Johnston, Kelly McGarel, Stephanie Feutren-Burton, Hendrik W. Van Den Berg, Timothy Mills, William Watters, Owen McGrath
Publikováno v: Bioconjugate Chemistry. 20:1737-1751
In this paper, we report the synthesis and biological activity of a series of dihydroisocoumarin analogues conjugated with fatty acids, alcohols, or amines, of varying hydrocarbon chain length and degree of unsaturation, to the dihydroisocoumarins, k
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1667f879679630d98eb3c2e7cc8c31e8
https://doi.org/10.1021/bc900122g
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8
Spinal Brucellosis
Autor: C W C William Watters rd., Charles A. Reitman
Publikováno v: Spine. 27:E250-E252
Study design Case report. Objective To increase awareness of spinal brucellosis and discuss demographics, diagnosis, and treatment. Summary of background data Brucellosis is a rare cause of spinal infections in the United States, although there have
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9000c01b5f81aa8a3437076c7e8e60d1
https://doi.org/10.1097/00007632-200205010-00028
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9
Abstract A175: Isolation and identification of compounds from the fruits of Kigelia pinnata with anti-proliferative activity towards human cancer cells
Autor: Stephanie Feutren-Burton, Paul Armstrong, Zoicha Delbederi, William Watters, Kelly McGarel, Hendrik W. Van Den Berg, Catherine A. Higgins, Owen McGrath, David Waugh
Publikováno v: Molecular Cancer Therapeutics. 8:A175-A175
Kigelia pinnata DC. (Bignoniaceae also referred to as K. Africana or sausage tree), is a tree which is found widely in Africa and the tropics in general. Traditionally hot aqueous extracts of fruit pods from Kigelia pinnata have been claimed to have
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::6101fd39f4d7b88983b75955d063228d
https://doi.org/10.1158/1535-7163.targ-09-a175
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10
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