Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Vishal Koradia"'
Publikováno v:
Pharmaceutics, Vol 4, Iss 1, Pp 93-103 (2012)
Amlodipine besilate, a calcium channel antagonist, exists in several solid forms. Processing of anhydrate and dihydrate forms of this drug may lead to solid state changes, and is therefore the focus of this study. Milling was performed for the anhydr
Externí odkaz:
https://doaj.org/article/adf55a3e3ebf450697a3d81313569125
Autor:
Lan Chen, Jagannath Kota, Vishal Koradia, Gangadhar Sunkara, Marie-Christine Wolf, Sampath Kalluri, F. Joel Leong, Daniel S. Stein, Jay Prakash Jain
Publikováno v:
Antimicrobial Agents and Chemotherapy
The artemether-lumefantrine combination requires food intake for the optimal absorption of lumefantrine. In an attempt to enhance the bioavailability of lumefantrine, new solid dispersion formulations (SDF) were developed, and the pharmacokinetics of
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0425d79536cf95188522f8943f10fca0
https://pubmed.ncbi.nlm.nih.gov/28630183
https://pubmed.ncbi.nlm.nih.gov/28630183
Publikováno v:
Pharmaceutics
Pharmaceutics, Vol 4, Iss 1, Pp 93-103 (2012)
Pharmaceutics; Volume 4; Issue 1; Pages: 93-103
Pharmaceutics, Vol 4, Iss 1, Pp 93-103 (2012)
Pharmaceutics; Volume 4; Issue 1; Pages: 93-103
Amlodipine besilate, a calcium channel antagonist, exists in several solid forms. Processing of anhydrate and dihydrate forms of this drug may lead to solid state changes, and is therefore the focus of this study. Milling was performed for the anhydr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::45cdc732ba323d3103c8fabd6f0f8fac
https://doi.org/10.3390/pharmaceutics4010093
https://doi.org/10.3390/pharmaceutics4010093
Autor:
Michiel Ringkjøbing-Elema, Heidi Lopez de Diego, Jørn Møller-Sonnergaard, Mikko Tenho, Jarno Salonen, Vishal Koradia, Vesa-Pekka Lehto, Jukka Rantanen
Publikováno v:
Pharmaceutical Research. 29:134-144
To investigate solid state transformations of drug substances during compaction using grazing incidence X-ray diffraction (GIXD). The solid forms of three model drugs–theophylline (TP), nitrofurantoin (NF) and amlodipine besylate (AMB)–were compa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fc9b52fdec3b6ce8b020376e8c08495c
https://doi.org/10.1007/s11095-011-0520-8
https://doi.org/10.1007/s11095-011-0520-8
Autor:
Jukka Rantanen, Claus Cornett, Vishal Koradia, Marja Savolainen, Fang Tian, Anette Müllertz, Johan Boetker, Thomas Rades, Jesper Østergaard
Publikováno v:
Molecular Pharmaceutics. 8:1372-1380
Traditional dissolution testing determines drug release to the bulk, but does not enable an understanding of the events happening close to the surface of a solid or a tablet. UV imaging is a new imaging approach that can be used to study the dissolut
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c085af62c8152d7ec0e88ae6d8385a63
https://doi.org/10.1021/mp200205z
https://doi.org/10.1021/mp200205z
Publikováno v:
Journal of Pharmaceutical Sciences. 99:3966-3976
There is a need for thorough knowledge of solid-state transformations in order to implement quality by design (QbD) methodology in drug development. The present study was aimed at gaining a mechanistic understanding of the dehydration of nitrofuranto
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8b4e6fecf1447da6e23e8e4b8d08c5df
https://doi.org/10.1002/jps.22244
https://doi.org/10.1002/jps.22244
Autor:
Jaakko Aaltonen, Vishal Koradia, Keith C. Gordon, Jukka Rantanen, Sabiruddin Mirza, Morten Allesø
Publikováno v:
European Journal of Pharmaceutics and Biopharmaceutics. 71:23-37
Solid form screening, the activity of generating and analysing different solid forms of an active pharmaceutical ingredient (API), has become an essential part of drug development. The multi-step screening process needs to be designed, performed and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c65d4b63e7eb097ec13d8161bc56014a
https://doi.org/10.1016/j.ejpb.2008.07.014
https://doi.org/10.1016/j.ejpb.2008.07.014
Publikováno v:
Excipient Applications in Formulation Design and Drug Delivery ISBN: 9783319202051
Generic drug products are defined as drug products that are comparable to the innovator/reference listed drug products (RLD) in dosage form, strength, route of administration, quality and performance characteristics, and intended use. These products
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4a925c25c1f9a905b2d650e133c7c8dd
https://doi.org/10.1007/978-3-319-20206-8_17
https://doi.org/10.1007/978-3-319-20206-8_17
Publikováno v:
Journal of Generic Medicines: The Business Journal for the Generic Medicines Sector. 2:335-346
Generic products are cost effective and speedy surrogates for high-priced innovator/branded products. The prerequisite for the development of a generic product is therapeutic equivalence (comprising pharmaceutical equivalence and bioequivalence) to t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0501f2efd27a93a86293e99bb9ee9fc2
https://doi.org/10.1057/palgrave.jgm.4940086
https://doi.org/10.1057/palgrave.jgm.4940086
Publikováno v:
Acta crystallographica. Section C, Crystal structure communications. 69(Pt 11)
Gaboxadol hydrochloride, also known as THIP hydrochloride (systematic name: 3-hydroxy-4,5,6,7-tetrahydro-1,2-oxazolo[5,4-c]pyridin-6-ium chloride), C6H9N2O2+·Cl−, exists as two enantiotropically related polymorphs. Transformation between the polym
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f91acb155734b26204bf160dbcf1a3bb
https://pubmed.ncbi.nlm.nih.gov/24192165
https://pubmed.ncbi.nlm.nih.gov/24192165