Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Vincenzo Proietto"'
Autor:
Xavier, Emonds-Alt, Vincenzo, Proietto, Régis, Steinberg, Florence, Oury-Donat, Xavier, Vigé, Pol, Vilain, Emmanuel, Naline, Samira, Daoui, Charles, Advenier, Gérard, Le Fur, Jean-Pierre, Maffrand, Philippe, Soubrié, Marc, Pascal
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 303:1171-1179
The biochemical and pharmacological properties of a novel antagonist of the tachykinin neurokinin 1 (NK1) receptor, SSR240600 [(R)-2-(1-[2-[4-[2-[3,5-bis(trifluoromethyl)phenyl]acetyl]-2-(3,4-dichlorophenyl)-2-morpholinyl]ethyl]-4-piperidinyl)-2-meth
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b7cd2c438709cbab96f371cd6ecfcedc
https://doi.org/10.1124/jpet.102.040162
https://doi.org/10.1124/jpet.102.040162
Autor:
Emmanuel Naline, Samira Daoui, Christiane Gueudet, Marc Pascal, Philippe Soubrie, Jean-Pierre Maffrand, Xavier Emonds-Alt, J.-C Michaud, Martine Poncelet, Gérard Le Fur, Régis Steinberg, Vincenzo Proietto, P. Vilain, Charles Advenier, F. Oury-Donat
Publikováno v:
Canadian Journal of Physiology and Pharmacology. 80:482-488
SSR 146977 is a potent and selective antagonist of the tachykinin NK3 receptor. In Chinese hamster ovary cells expressing the human tachykinin NK3 receptor, SSR 146977 inhibited the binding of radioactive neurokinin B to NK3 receptors (Ki = 0.26 nM),
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2bdb1d3396507e9e8e44b44e1299ca6d
https://doi.org/10.1139/y02-041
https://doi.org/10.1139/y02-041
Autor:
G. Le Fur, S Daoul, J.C. Brelière, D. Van Broeck, M. Poncelet, Charles Advenier, Jean-Philippe Ducoux, Marco Landi, Emmanuel Naline, C Cognon, Philippe Soubrie, Vincenzo Proietto, X. Emonds-Alt, P. Vilain, Gervais Neliat, J P Maffrand, T. Croci
Publikováno v:
Neuropeptides. 31:449-458
(R)-3-(1-[2-(4-benzoyl-2-(3,4-difluorophenyl)-morpholin-2-yl)- ethyl]-4-phenylpiperidin-4-yl)-1-dimethylurea (SR 144190) is a new non-peptide antagonist of tachykinin NK2 receptors. SR 144190 potently and selectively inhibited neurokinin A binding to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::635453df0e79e08dfa3ea9112dc64bd6
https://doi.org/10.1016/s0143-4179(97)90039-1
https://doi.org/10.1016/s0143-4179(97)90039-1
Autor:
Daniel Bichon, B. Miloux, M. Poncelet, J.C. Brele`ere, Gervais Neliat, X. Emonds-Alt, Jean-Philippe Ducoux, Vincenzo Proietto, P. Vilain, D. Van Broeck, Michel Heaulme, Philippe Soubrie, G. Le Fur
Publikováno v:
Life Sciences. 56:PL27-PL32
SR 142801 is the first potent and selective non-peptide antagonist of the tachykinin NK3 receptor. It inhibited [MePhe7]NKB binding to its receptor from various species, including humans. SR 142801 was a competitive antagonist of [MePhe7]NKB-mediated
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::00cba3ece7eda5bf9198e2c8b7ed1fc4
https://doi.org/10.1016/0024-3205(94)00413-m
https://doi.org/10.1016/0024-3205(94)00413-m
Autor:
Vincenzo Proietto, Gervais Neliat, P. Vilain, Jean-Philippe Ducoux, Jean-Daniel Doutremepuich, Régis Steinberg, Philippe Soubrie, Xavier Emonds-Alt, Michel Heaulme, Gérard Le Fur, Didier Van Broeck, Jean-Claude Breliere, Vincent Santucci, Daniel Bichon
Publikováno v:
European Journal of Pharmacology. 250:403-413
(S)1-(2-[3-(3,4-dichlorophenyl)-1-(3-isopropoxyphenylacetyl)pip eridin-3- yl]ethyl)-4-phenyl-1-azoniabicyclo[2.2.2]octane chloride (SR140333) is a new non-peptide antagonist of tachykinin NK1 receptors. SR140333 potently, selectively and competitivel
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a2fb1e52b6a1f357aee3e05caa5d8387
https://doi.org/10.1016/0014-2999(93)90027-f
https://doi.org/10.1016/0014-2999(93)90027-f
Autor:
Vincent Santucci, Xavier Emonds-Alt, Didier Van Broeck, Gervais Neliat, Vincenzo Proietto, P. Vilain, Jean-Claude Breliere, Luciano Manara, Gérard Le Fur, Charles Advenier, Philippe Soubrie, T. Croci, Martine Poncelet
Publikováno v:
Regulatory Peptides. 46:31-36
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::abd725b81e75a1c6a8b55af239805131
https://doi.org/10.1016/0167-0115(93)90008-v
https://doi.org/10.1016/0167-0115(93)90008-v
Autor:
Emmanuel Naline, Pierre Yves Andre Goulaouic, J.C. Brelière, G. Le Fur, D. Van Broeck, Gervais Neliat, Vincenzo Proietto, P. Vilain, Charles Advenier, X. Emonds-Alt
Publikováno v:
Life sciences. 50(15)
SR 48968 is a potent and selective non-peptide antagonist of the neurokinin A (NK2) receptor. SR 48968 selectively inhibited neurokinin A binding to its receptor and was a competitive antagonist of neurokinin A-mediated contraction of different isola
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c15442fe8520c5e9a040933080ccb7df
https://pubmed.ncbi.nlm.nih.gov/1313515
https://pubmed.ncbi.nlm.nih.gov/1313515
Autor:
Gervais Neliat, J.C. Brelière, X. Emonds-Alt, D. Van Broeck, Vincenzo Proietto, P. Vilain, Pierre Yves Andre Goulaouic, Emmanuel Naline, Charles Advenier, G Le Fur
Publikováno v:
Neuropeptides. 22:21-22
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::2dce91d53279fdbc19c830ff77bc195f
https://doi.org/10.1016/0143-4179(92)90392-a
https://doi.org/10.1016/0143-4179(92)90392-a