Zobrazeno 1 - 10
of 20
pro vyhledávání: '"Vincent Remusat"'
Publikováno v:
The Journal of Organic Chemistry. 87:4483-4488
We describe herein the intermolecular addition reaction of benzyl halides to aldehydes and imines using photoactivated tetrakis(dimethylamino)ethylene (TDAE) as superphotoreductant. 3,4-Dihydroisocoumarins, 1,2-diarylethanols, and 1,2-diarylcarbamate
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ab88b54676a4835fc20ff78cc232bd01
https://doi.org/10.1021/acs.joc.2c00074
https://doi.org/10.1021/acs.joc.2c00074
Autor:
Pierre Verhaeghe, Nadine Azas, Vincent Remusat, Armand Gellis, Sébastien Hutter, Gilles Lanzada, Nicolas Primas, Patrice Vanelle
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 2016, 119, pp.34-44. ⟨10.1016/j.ejmech.2016.04.059⟩
European Journal of Medicinal Chemistry, 2016, 119, pp.34-44. ⟨10.1016/j.ejmech.2016.04.059⟩
European Journal of Medicinal Chemistry, Elsevier, 2016, 119, pp.34-44. ⟨10.1016/j.ejmech.2016.04.059⟩
European Journal of Medicinal Chemistry, 2016, 119, pp.34-44. ⟨10.1016/j.ejmech.2016.04.059⟩
International audience; A DMAP catalyzedsynthesis of new 4-benzyloxy-and 4-aryloxy-2-trichloromethylquinazolines was studied, in a view to react 4-chloroquinazolines with poorly nucleophilic alcohols such as benzylic alcohols, via a simple and cheapS
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::42d8abb3ecaa18899fdd3bf692cff6a7
https://pubmed.ncbi.nlm.nih.gov/27155463
https://pubmed.ncbi.nlm.nih.gov/27155463
Autor:
Vincent Remusat, Patrice Vanelle, Nicolas Primas, Youssef Kabri, Christophe Curti, Clémence Tabélé
Publikováno v:
ChemInform. 47
To obtain aromatic 2-methylallyl derivatives, cross-coupling reactions between 2-methyl-2-propen-1-ol and various boronic acids were studied. Among allylic alcohols described for such cross-coupling reactions, 2-methyl-2-propen-1-ol has a low reactiv
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7b2afc2e79f9bb050f2765fd51099be9
https://doi.org/10.1002/chin.201610067
https://doi.org/10.1002/chin.201610067
Autor:
Pierre Verhaeghe, Caroline Castera-Ducros, J. C. Teulade, Melanie Piednoel, Vincent Remusat, Patrice Vanelle, Pascal Rathelot, Hussein El-Kashef
Publikováno v:
Letters in Organic Chemistry
Letters in Organic Chemistry, Bentham Science Publishers, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩
Letters in Organic Chemistry, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩
Letters in Organic Chemistry, Bentham Science Publishers, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩
Letters in Organic Chemistry, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩
International audience; Background:The imidazo[1,2-alpha] pyridine ring has been widely studied by medicinal chemists and displays great pharmaceutical potential. Methods: In a view to prepare a library of new molecules including an imidazo[1,2-alpha
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1e75b64d6b888be1ac4140ca49e6979d
https://hal.archives-ouvertes.fr/hal-01460673
https://hal.archives-ouvertes.fr/hal-01460673
Publikováno v:
Synthesis. 2009:3150-3156
A new simple, rapid and high yielding synthesis (mean yield = 83%) of various 4-aryl, 4-heteroaryl, and 4-styryl-1,2-dimethyl-5-nitro-1H-imidazoles by palladium-catalyzed Suzuki― Miyaura cross-coupling reactions using microwave irradiation is descr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7b1e64b35c01f89ec5edeed6d33d7a8c
https://doi.org/10.1055/s-0029-1216905
https://doi.org/10.1055/s-0029-1216905
Autor:
Nadine Azas, Céline Botta, Michel De Méo, Vincent Remusat, Monique Gasquet, Patrice Vanelle, Maxime D. Crozet, Sébastien Hutter, Christophe Curti, Olivier Chapelle
Publikováno v:
European Journal of Medicinal Chemistry. 44:653-659
To improve the antiparasitic pharmacophore, 20 5-nitroimidazoles bearing an arylsulfonylmethyl group were prepared from commercial imidazoles. The antiparasitic activity of these molecules was assessed against Trichomonas vaginalis, the in vitro cyto
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::41cb4a6042e647afa988c0797eeb2023
https://doi.org/10.1016/j.ejmech.2008.05.015
https://doi.org/10.1016/j.ejmech.2008.05.015
Autor:
Nicolas Primas, Vincent Remusat, Youssef Kabri, Clémence Tabélé, Patrice Vanelle, Christophe Curti
Publikováno v:
Synthesis: Journal of Synthetic Organic Chemistry
Synthesis: Journal of Synthetic Organic Chemistry, 2015, 47, pp.3339-3346. ⟨10.1055/s-0034-1381034⟩
SYNTHESIS
SYNTHESIS, Georg Thieme Verlag, 2015, 47, pp.3339-3346. ⟨10.1055/s-0034-1381034⟩
Synthesis: Journal of Synthetic Organic Chemistry, 2015, 47, pp.3339-3346. ⟨10.1055/s-0034-1381034⟩
SYNTHESIS
SYNTHESIS, Georg Thieme Verlag, 2015, 47, pp.3339-3346. ⟨10.1055/s-0034-1381034⟩
International audience; To obtain aromatic 2-methylallyl derivatives, cross-coupling reactions between 2-methyl-2-propen-1-ol and various boronic acids were studied. Among allylic alcohols described for such cross-coupling reactions, 2-methyl-2-prope
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c0865ba64332f72df0f15ca9a57bcae1
https://hal.science/hal-01423338/document
https://hal.science/hal-01423338/document
Autor:
Patrice Vanelle, Sylvain Rault, Charline Kieffer, Pascal Rathelot, Anita Cohen, Caroline Castera-Ducros, Nadine Azas, Pierre Verhaeghe, Sébastien Hutter, Manel Kraiem M'Rabet, Michèle Laget, Vincent Remusat
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, 2015, 92, pp.282-294. ⟨10.1016/j.ejmech.2014.12.056⟩
European Journal of Medicinal Chemistry, Elsevier, 2015, 92, pp.282--294. 〈10.1016/j.ejmech.2014.12.056〉
European Journal of Medicinal Chemistry, Elsevier, 2015, 92, pp.282-294. ⟨10.1016/j.ejmech.2014.12.056⟩
European Journal of Medicinal Chemistry, 2015, 92, pp.282-294. ⟨10.1016/j.ejmech.2014.12.056⟩
European Journal of Medicinal Chemistry, Elsevier, 2015, 92, pp.282--294. 〈10.1016/j.ejmech.2014.12.056〉
European Journal of Medicinal Chemistry, Elsevier, 2015, 92, pp.282-294. ⟨10.1016/j.ejmech.2014.12.056⟩
International audience; From a recently identified antileishmanial pharmacophore, a structure activity relationship study was conducted by introducing various aminated, phenoxy or thiophenoxy moieties at position 4 of the 8-nitroquinolin-2(1H)-one sc
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c2609075b515fa1892285b6a4c9336d3
https://hal-amu.archives-ouvertes.fr/hal-01460569
https://hal-amu.archives-ouvertes.fr/hal-01460569
Publikováno v:
Synthetic Communications. 36:3639-3646
Original 4‐arylsulfonylmethyl‐5‐nitroimidazoles were prepared by reacting four chloromethylaryl sulfones with 5‐nitroimidazole derivatives via a vicarious nucleophilic substitution (VNS) of hydrogen reaction.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::63b56932d59f48866fba61b33669420e
https://doi.org/10.1080/00397910600943873
https://doi.org/10.1080/00397910600943873
Publikováno v:
Journal of Heterocyclic Chemistry. 41:221-225
A new heterocyclic bioreductive bis-alkylating agent, 2,3-bis(chloromethyl)benzo[g]quinoxaline-5,10-dione, was prepared in a four-steps synthesis. It was shown to react under electron transfer conditions with 2-nitropropane anion by an bis-SRN1 mecha
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ed28f4368496f52c10ea79bc6d570f01
https://doi.org/10.1002/jhet.5570410212
https://doi.org/10.1002/jhet.5570410212