Výsledky vyhledávání - "Vijay M. Prajapati"

One-Pot Synthesis of 3,4-Diaryl-Substituted 2(5H)-Furanone and Its Commercial Application

Autor: Anil Argade, Pravin Thombare, Mukul R. Jain, Sanjay Gite, Vijay M. Prajapati, Jigar Desai, Kiran Shah, Pankaj R. Patel, Bipin Pandey, Rajesh Bahekar

Publikováno v: Synthetic Communications. 42:3140-3149

One-pot synthesis of 3,4-diaryl substituted 2(5H)-furanones was established and its commercial application has been demonstrated by accomplishing total synthesis of rofecoxib, under mild reaction conditions, with good yields and purity.

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::e1c8e11aa3d9d51d929cf9953cd9d66b
https://doi.org/10.1080/00397911.2011.577923

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An improved synthesis of Fmoc-N-methyl serine and threonine

Autor: Arun A. Gupta, Rajesh H. Bahekar, Dipam Patel, Pankaj R. Patel, Vijay M. Prajapati, Pradip Jadav, Mukul R. Jain

Publikováno v: Tetrahedron Letters. 48:5003-5005

An improved method for the synthesis of Fmoc-N-methyl serine and threonine has been developed, which involves formation and subsequent reduction of the corresponding oxazolidinone with a Lewis acid under mild conditions, with improved yields and shor

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::55ea938c6ebbb4cfbd37d131b18a30a5
https://doi.org/10.1016/j.tetlet.2007.05.112

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Synthesis and antidiabetic activity of 2,5-disubstituted-3-imidazol-2-yl-pyrrolo[2,3-b]pyridines and thieno[2,3-b]pyridines

Autor: Honey Modi, Mukul R. Jain, Pankaj R. Patel, Arun A. Gupta, Rajesh H. Bahekar, Dipam Patel, Ajay Sharma, Pradip Jadav, Vijay M. Prajapati, Debdutta Bandyopadhya, Robby Tom

Publikováno v: Bioorganicmedicinal chemistry. 15(21)

In the present investigation, two series of 2,5-disubstituted-3-imidazol-2-yl-pyrrolo[2,3-b]pyridines (2a–l) and thieno[2,3-b]pyridines (3a–l) were designed as analogs of BL 11282 (1). The in vitro glucose dependent insulinotropic activity of all

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c2a247763420c106f89458a38ca9911e
https://pubmed.ncbi.nlm.nih.gov/17723306

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Synthesis of 3,8,9-trisubstituted-1,7,9-triaza-fluorene-6-carboxylic acid derivatives as a new class of insulin secretagogues

Autor: Arun A. Gupta, Ashish Goel, Pradip Jadav, Dipam Patel, Rajesh Bahekar, Pankaj R. Patel, Vijay M. Prajapati, Mukul R. Jain, Honey Modi

Publikováno v: Bioorganicmedicinal chemistry. 15(17)

beta-Carbolines stimulate insulin secretion in a glucose-dependent manner, probably by acting on I(3)-binding site. Knowing the in vitro glucose-dependent insulinotropic potential of beta-carbolines, in this project, three series of substituted-triaz

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a5f544fa55ca78f364819301182fa254
https://pubmed.ncbi.nlm.nih.gov/17583514

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Design, synthesis, and biological evaluation of substituted-N-(thieno[2,3-b]pyridin-3-yl)-guanidines, N-(1H-pyrrolo[2,3-b]pyridin-3-yl)-guanidines, and N-(1H-indol-3-yl)-guanidines

Autor: Arun A. Gupta, Ashish Goel, Mukul R. Jain, Dipam Patel, Pankaj R. Patel, Pradip Jadav, Rajesh Bahekar, Vijay M. Prajapati

Publikováno v: Bioorganicmedicinal chemistry. 15(9)

Sulfonylureas stimulate insulin secretion independent of the blood glucose concentration and therefore cause hypoglycemia in type 2 diabetic patients. Over the last years, a number of aryl-imidazoline derivatives have been identified that stimulate i

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58ee9b0ff6b95a35036f1a896e68049f
https://pubmed.ncbi.nlm.nih.gov/17339113

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